Full Name
Tafi, Andrea
 
DBCF community
 
Discipline (SSD)
CHIM/08 - Chimica Farmaceutica
 
Email UNISI
andrea.tafi@unisi.it
 
 
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Publications
(Articles)



Results 1-20 of 82 (Search time: 0.009 seconds).

Issue DateTitleAuthor(s)Third Mission
120081-[(3-Aryloxy-3-aryl)propyl]-2H-imidazoles, new imidazoles with potent activity against Candida albicans and dermatophytes. Synthesis, structure-activity relationship, and molecular modeling studiesG., LA REGINA; F., D'Auria; Tafi, Andrea ; F., Piscitelli; S., Olla; F., Caporuscio; L., Nencioni; R., Cirilli; F., LA TORRE; N., RODRIGUES DE MELO; S., Kelly; D., Lamb; M., Artico; Botta, Maurizio ; A., Palamara; R., SilvestriNot applicable
220133D-QSAR using pharmacophore-based alignment and virtual screening for discovery of novel MCF-7 cell line inhibitorsBrogi, Simone; Panagiota, Papazafiri; Vassilios, Roussis; Tafi, Andrea Not applicable
32002Alpha1-Adrenoceptor Antagonists. 4. Pharmacophore-based Design, Synthesis, and Biological Evaluation of New Imidazo-, Benzimidazo-, and Indoloarylpiperazine DerivativesL., Betti; Botta, Maurizio ; Corelli, Federico ; S., Corsano; M., Floridi; G., Giannaccini; L., Maccari; Manetti, Fabrizio ; G., Strappaghetti; Tafi, Andrea Not applicable
42005AMBER force field implementation of the boronate function to simulate the inhibition of β-lactamases by alkyl and aryl boronic acids.Tafi, Andrea ; M., Agamennone; P., Tortorella; S., Alcaro; C., Gallina; Botta, Maurizio Not applicable
52002Antifungal agents. 10. New derivatives of 1-[(Aryl)[4-aryl-1H-pyrrol-3-yl]methyl]-1H-imidazole, synthesis, anti-Candida activity and Quantitative Structure-Analysis Relationship studiesTafi, Andrea ; R., Costi; Botta, Maurizio ; R., DI SANTO; Corelli, Federico ; Massa, Silvio; A., Ciacci; Manetti, Fabrizio ; M., ArticoNot applicable
62005Antifungal Agents. 11.N-Substituted Derivatives of 1-[(Aryl)(4-aryl-1H-pyrrol-3yl)methyl]-1H-imidazole: Synthesis, Anti-Candida Activity, and QSAR StudiesDi Santo, Roberto; Tafi, Andrea ; Costi, Roberta; Botta, Maurizio ; Artico, Marino; Corelli, Federico ; Forte, Michela; Caporuscio, Fabiana; Angiolella, Letizia; Palamara, Anna TeresaNot applicable
72004Antimycobacterial compounds. New pyrrole derivatives of BM212Biava, M.; Porretta, G. C.; Deidda, D.; Pompei, R.; Tafi, Andrea ; Manetti, Fabrizio Not applicable
82005Antimycobacterial compounds. Optimization of the BM212 structure, the lead compound for a new pyrrole derivative classBiava, M; Porretta, Gc; Poce, G; Deidda, D; Pompei, R; Tafi, Andrea ; Manetti, Fabrizio Not applicable
92007An approach to address Candida rugosa lipase regioselectivity in the acylation reactions of trytilated glucosidesC., Palocci; M., Falconi; S., Alcaro; Tafi, Andrea ; R., Puglisi; F., Ortuso; Botta, Maurizio ; L., Alberghina; E., CerniaNot applicable
102007Bis(diamido)-bridged basket resorcin[4]arenes as enantioselective receptors for amino acids and aminesBotta, B; D'Acquarica, F; Nevola, L; Sacco, F; Lopez, Zv; Zappia, G; Fraschetti, C; Speranza, M; Tafi, Andrea ; Caporuscio, F; Letzel, Mc; Mattay, J.Not applicable
112004Cavity Effects on the Enantioselectivity of Chiral Amido[4]resorcinarene StereoisomersB., Botta; D., Subissati; Tafi, Andrea ; G., DELLE MONACHE; A., Filippi; M., SperanzaNot applicable
122001Chair-boat equilibrium as driving force in epimerization of 3,7-dimethylbicyclo[3.3.1]nonan-2,9-dione derivatives. Stereocontrolled synthesis of 3-exo,7-exo- and 3-endo,7-exo-3,7-dimethylbicyclo[3.3.1]nonan-9-onesA., Gambacorta; D., Tofani; Tafi, Andrea ; M., ELMI FARAHNot applicable
132004Chalcone Prenyltransferase from Morus nigra cell cultures. Substrate specificity studiesVitali, A.; Botta, B.; Tafi, Andrea ; Silvestrini, A.; DELLE MONACHE, G.; Giardina, B.; Rocca, F.Not applicable
142012Characterization of COR627 and COR628, two novel positive allosteric modulators of the GABA B receptorCastelli, M. P.; Casu, A.; Casti, P.; Lobina, C.; Carai, M. A. M.; Colombo, G.; Solinas, M.; Giunta, D.; Mugnaini, Claudia ; Pasquini, Serena; Tafi, Andrea ; Brogi, Simone; Gessa, G. L.; Corelli, Federico Not applicable
152004Chiral Recognition by Resorcin[4]arene Receptors: Intrinsic Kinetics and DynamicsTafi, Andrea ; Bruno, Botta; Botta, Maurizio ; GIULIANO DELLE, Monache; Antonello, Filippi; Maurizio, SperanzaNot applicable
162006Computational studies of competitive inhibitors of nitric oxide synthase (NOS) enzymes: towards the development of powerful and isoform-selective inhibitors.Tafi, Andrea ; Angeli, Lucilla; Venturini, G; Travagli, Massimiliano; Corelli, Federico ; Botta, Maurizio Not applicable
172000Computer Simulations of Enantioselective Ester Hydrolyses Catalyzed by Pseudomonas cepacia LipaseTafi, Andrea ; Van Almsick, Andreas; Corelli, Federico ; Crusco, Maria; Laumen Kurt, E.; Schneider Manfred, P.; Botta, Maurizio Not applicable
181992CONFORMATIONAL EFFECTS ON THE STEREOCHEMICAL COURSE OF THE NABH4 REDUCTION OF SUBSTITUTED BICYCLO[3.3.1]NONAN-2-ONESGambacorta, A; Dellojacono, Ar; Botta, Maurizio ; Tafi, Andrea Not applicable
192001Conformational search of antisense nucleotidesStefano, Alcaro; Tafi, Andrea ; Francesco, Ortuso; Lucyna A., Woźniak; Eszter Gács, Baitz; Botta, Maurizio Not applicable
202004Conformational search of antisense nucleotides. Part. 2Alcaro, S; Ortuso, F; Gallelli, A; Battaglia, D; Tafi, Andrea ; Botta, Maurizio Not applicable