Tafi, Andrea
Claim profile
Full Name
Tafi, Andrea
DBCF community
Discipline (SSD)
CHIM/08 - Chimica Farmaceutica
Email UNISI
andrea.tafi@unisi.it





Publications
(Articles)
Results 1-20 of 82 (Search time: 0.009 seconds).
Issue Date | Title | Author(s) | Third Mission | |
---|---|---|---|---|
1 | 2008 | 1-[(3-Aryloxy-3-aryl)propyl]-2H-imidazoles, new imidazoles with potent activity against Candida albicans and dermatophytes. Synthesis, structure-activity relationship, and molecular modeling studies | G., LA REGINA; F., D'Auria; Tafi, Andrea ; F., Piscitelli; S., Olla; F., Caporuscio; L., Nencioni; R., Cirilli; F., LA TORRE; N., RODRIGUES DE MELO; S., Kelly; D., Lamb; M., Artico; Botta, Maurizio ; A., Palamara; R., Silvestri | Not applicable |
2 | 2013 | 3D-QSAR using pharmacophore-based alignment and virtual screening for discovery of novel MCF-7 cell line inhibitors | Brogi, Simone; Panagiota, Papazafiri; Vassilios, Roussis; Tafi, Andrea | Not applicable |
3 | 2002 | Alpha1-Adrenoceptor Antagonists. 4. Pharmacophore-based Design, Synthesis, and Biological Evaluation of New Imidazo-, Benzimidazo-, and Indoloarylpiperazine Derivatives | L., Betti; Botta, Maurizio ; Corelli, Federico ; S., Corsano; M., Floridi; G., Giannaccini; L., Maccari; Manetti, Fabrizio ; G., Strappaghetti; Tafi, Andrea | Not applicable |
4 | 2005 | AMBER force field implementation of the boronate function to simulate the inhibition of β-lactamases by alkyl and aryl boronic acids. | Tafi, Andrea ; M., Agamennone; P., Tortorella; S., Alcaro; C., Gallina; Botta, Maurizio | Not applicable |
5 | 2002 | Antifungal agents. 10. New derivatives of 1-[(Aryl)[4-aryl-1H-pyrrol-3-yl]methyl]-1H-imidazole, synthesis, anti-Candida activity and Quantitative Structure-Analysis Relationship studies | Tafi, Andrea ; R., Costi; Botta, Maurizio ; R., DI SANTO; Corelli, Federico ; Massa, Silvio; A., Ciacci; Manetti, Fabrizio ; M., Artico | Not applicable |
6 | 2005 | Antifungal Agents. 11.N-Substituted Derivatives of 1-[(Aryl)(4-aryl-1H-pyrrol-3yl)methyl]-1H-imidazole: Synthesis, Anti-Candida Activity, and QSAR Studies | Di Santo, Roberto; Tafi, Andrea ; Costi, Roberta; Botta, Maurizio ; Artico, Marino; Corelli, Federico ; Forte, Michela; Caporuscio, Fabiana; Angiolella, Letizia; Palamara, Anna Teresa | Not applicable |
7 | 2004 | Antimycobacterial compounds. New pyrrole derivatives of BM212 | Biava, M.; Porretta, G. C.; Deidda, D.; Pompei, R.; Tafi, Andrea ; Manetti, Fabrizio | Not applicable |
8 | 2005 | Antimycobacterial compounds. Optimization of the BM212 structure, the lead compound for a new pyrrole derivative class | Biava, M; Porretta, Gc; Poce, G; Deidda, D; Pompei, R; Tafi, Andrea ; Manetti, Fabrizio | Not applicable |
9 | 2007 | An approach to address Candida rugosa lipase regioselectivity in the acylation reactions of trytilated glucosides | C., Palocci; M., Falconi; S., Alcaro; Tafi, Andrea ; R., Puglisi; F., Ortuso; Botta, Maurizio ; L., Alberghina; E., Cernia | Not applicable |
10 | 2007 | Bis(diamido)-bridged basket resorcin[4]arenes as enantioselective receptors for amino acids and amines | Botta, B; D'Acquarica, F; Nevola, L; Sacco, F; Lopez, Zv; Zappia, G; Fraschetti, C; Speranza, M; Tafi, Andrea ; Caporuscio, F; Letzel, Mc; Mattay, J. | Not applicable |
11 | 2004 | Cavity Effects on the Enantioselectivity of Chiral Amido[4]resorcinarene Stereoisomers | B., Botta; D., Subissati; Tafi, Andrea ; G., DELLE MONACHE; A., Filippi; M., Speranza | Not applicable |
12 | 2001 | Chair-boat equilibrium as driving force in epimerization of 3,7-dimethylbicyclo[3.3.1]nonan-2,9-dione derivatives. Stereocontrolled synthesis of 3-exo,7-exo- and 3-endo,7-exo-3,7-dimethylbicyclo[3.3.1]nonan-9-ones | A., Gambacorta; D., Tofani; Tafi, Andrea ; M., ELMI FARAH | Not applicable |
13 | 2004 | Chalcone Prenyltransferase from Morus nigra cell cultures. Substrate specificity studies | Vitali, A.; Botta, B.; Tafi, Andrea ; Silvestrini, A.; DELLE MONACHE, G.; Giardina, B.; Rocca, F. | Not applicable |
14 | 2012 | Characterization of COR627 and COR628, two novel positive allosteric modulators of the GABA B receptor | Castelli, M. P.; Casu, A.; Casti, P.; Lobina, C.; Carai, M. A. M.; Colombo, G.; Solinas, M.; Giunta, D.; Mugnaini, Claudia ; Pasquini, Serena; Tafi, Andrea ; Brogi, Simone; Gessa, G. L.; Corelli, Federico | Not applicable |
15 | 2004 | Chiral Recognition by Resorcin[4]arene Receptors: Intrinsic Kinetics and Dynamics | Tafi, Andrea ; Bruno, Botta; Botta, Maurizio ; GIULIANO DELLE, Monache; Antonello, Filippi; Maurizio, Speranza | Not applicable |
16 | 2006 | Computational studies of competitive inhibitors of nitric oxide synthase (NOS) enzymes: towards the development of powerful and isoform-selective inhibitors. | Tafi, Andrea ; Angeli, Lucilla; Venturini, G; Travagli, Massimiliano; Corelli, Federico ; Botta, Maurizio | Not applicable |
17 | 2000 | Computer Simulations of Enantioselective Ester Hydrolyses Catalyzed by Pseudomonas cepacia Lipase | Tafi, Andrea ; Van Almsick, Andreas; Corelli, Federico ; Crusco, Maria; Laumen Kurt, E.; Schneider Manfred, P.; Botta, Maurizio | Not applicable |
18 | 1992 | CONFORMATIONAL EFFECTS ON THE STEREOCHEMICAL COURSE OF THE NABH4 REDUCTION OF SUBSTITUTED BICYCLO[3.3.1]NONAN-2-ONES | Gambacorta, A; Dellojacono, Ar; Botta, Maurizio ; Tafi, Andrea | Not applicable |
19 | 2001 | Conformational search of antisense nucleotides | Stefano, Alcaro; Tafi, Andrea ; Francesco, Ortuso; Lucyna A., Woźniak; Eszter Gács, Baitz; Botta, Maurizio | Not applicable |
20 | 2004 | Conformational search of antisense nucleotides. Part. 2 | Alcaro, S; Ortuso, F; Gallelli, A; Battaglia, D; Tafi, Andrea ; Botta, Maurizio | Not applicable |