Full Name
Gemma, Sandra
 
DBCF community
 
Discipline (SSD)
CHIM/08 - Chimica Farmaceutica
 
Email UNISI
sandra.gemma@unisi.it
 
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Publications
(Articles)

Results 1-20 of 117 (Search time: 0.004 seconds).

Issue DateTitleAuthor(s)Third Mission
120081H-Cyclopentapyrimidine-2,4(1H,3H)-dione-Related Ionotropic Glutamate Receptors Ligands. Structure-Activity Relationships and Identification of Potent and Selective iGluR5 ModulatorsButini, Stefania ; DARRYL S., Pickering; Elena, Morelli; SANNA COCCONE, Salvatore; Trotta, Francesco; MERI DE, Angelis; Guarino, Egeria; Fiorini, Isabella; Campiani, Giuseppe ; Ettore, Novellino; Arne, Schousboe; JEPPE K., Christensen; Gemma, Sandra Not applicable
22017Activation of the Wnt pathway by small peptides: rational design, synthesis and biological evaluationBrogi, Simone; Maramai, Samuele ; Brindisi, Margherita ; Chemi, Giulia ; Porcari, Valentina; Corallo, Claudio; Gennari, Luigi; Novellino, Ettore; Ramunno, Anna; Butini, Stefania ; Campiani, Giuseppe ; Gemma, Sandra Not applicable
32018Antimalarial agents against both sexual and asexual parasites stages: structure-activity relationships and biological studies of the Malaria Box compound 1-[5-(4-bromo-2-chlorophenyl)furan-2-yl]- N -[(piperidin-4-yl)methyl]methanamine (MMV019918) and analoguesVallone, Alessandra; D'Alessandro, Sarah; Brogi, Simone; Brindisi, Margherita ; Chemi, Giulia ; Alfano, Gloria; Lamponi, Stefania ; Lee, Soon Goo; Jez, Joseph M.; Koolen, Karin J. M.; Dechering, Koen J.; Saponara, Simona; Fusi, Fabio ; Gorelli, Beatrice; Taramelli, Donatella; Parapini, Silvia; Caldelari, Reto; Campiani, Giuseppe ; Gemma, Sandra ; Butini, Stefania Not applicable
42016Antitumor effect of pyrrolo-1,5-benzoxazepine-15 and its synergistic effect with Oxaliplatin and 5-FU in colorectal cancer cellsFiore, Donatella; Proto, Maria Chiara; Pisanti, Simona; Picardi, Paola; Pagano Zottola, Antonio Christian; Butini, Stefania ; Gemma, Sandra ; Casagni, Alice; Laezza, Chiara; Vitale, Mario; Ligresti, Alessia; Di Marzo, Vincenzo; Zisterer, Daniela M; Nathwani, Seema; Williams, D Clive; Campiani, Giuseppe ; Gazzerro, Patrizia; Bifulco, MaurizioNot applicable
52019Autophagy modulators for the treatment of oral and esophageal squamous cell carcinomasKhan, Tuhina ; Relitti, Nicola ; Brindisi, Margherita ; Magnano, S.; Zisterer, D.; Gemma, Sandra ; Butini, Stefania ; Campiani, Giuseppe Not applicable
62008Beta-secretase as a therapeutic target for Alzheimer’s diseaseA. K., Ghosh; Gemma, Sandra ; J., TangNot applicable
72019Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes-5Mangoni, Arduino A; Eynde, Jean Jacques Vanden; Jampilek, Josef; Hadjipavlou-Litina, Dimitra; Liu, Hong; Reynisson, Jóhannes; Sousa, Maria Emília; Gomes, Paula A C; Prokai-Tatrai, Katalin; Tuccinardi, Tiziano; Sabatier, Jean-Marc; Luque, F Javier; Rautio, Jarkko; Karaman, Rafik; Vasconcelos, M Helena; Gemma, Sandra ; Galdiero, Stefania; Hulme, Christopher; Collina, Simona; Gütschow, Michael; Kokotos, George; Siciliano, Carlo; Capasso, Raffaele; Agrofoglio, Luigi A; Ragno, Rino; Muñoz-Torrero, DiegoNot applicable
82019Bridged bicyclic 2,3-dioxabicyclo[3.3.1]nonanes as antiplasmodial agents: Synthesis, structure-activity relationships and studies on their biomimetic reaction with Fe(II)D'Alessandro, S.; Alfano, G.; Di Cerbo, L.; Brogi, S.; Chemi, Giulia ; Relitti, Nicola ; Brindisi, Margherita ; Lamponi, Stefania ; Novellino, E.; Campiani, Giuseppe ; Gemma, Sandra ; Basilico, N.; Taramelli, D.; Baratto, Maria Camilla ; Pogni, Rebecca ; Butini, Stefania Not applicable
92011Broad inhibition of plasmodium falciparum cytoadherence by (+)-epigallocatechin gallatePatil, PRADEEP RANGRAO; Gemma, Sandra ; Campiani, Giuseppe ; Alister G., CraigNot applicable
102011The Ca2+-ATPase (SERCA1) Is Inhibited by 4-Aminoquinoline Derivatives through Interference with Catalytic Activation by Ca2+, Whereas the ATPase E2 State Remains FunctionalG., Bartolommei; F., Tadini Buoninsegni; M. R., Moncelli; Gemma, Sandra ; Camodeca, Caterina; Butini, Stefania ; Campiani, Giuseppe ; D., Lewis; G., InesiNot applicable
112019Cinnamic acids derived compounds with antileishmanial activity target Leishmania amazonensis arginaseda Silva, Edson Roberto; Brogi, Simone; Grillo, Alessandro; Campiani, Giuseppe ; Gemma, Sandra ; Vieira, Paulo Cezar; Maquiaveli, Claudia do CarmoNot applicable
122008Clotrimazole Scaffold as an Innovative Pharmacophore Towards Potent Antimalarial Agents: Design, Synthesis, Biological and Structure-Activity Relationship Studies.Gemma, Sandra ; Campiani, Giuseppe ; Butini, Stefania ; G., Kukreja; SANNA COCCONE, Salvatore; B., Joshi; M., Persico; Nacci, Vito; Fiorini, Isabella; E., Novellino; Fattorusso, E; O., TAGLIALATELA SCAFATI; Savini, Luisa; D., Taramelli; N., Basilico; S., Parapini; G., Morace; V., Yardley; S., Croft; M., Coletta; S., Marini; Fattorusso, CaterinaNot applicable
132009Combining 4-Aminoquinoline- and Clotrimazole-based Pharmacophores towards Innovative and Potent Hybrid Antimalarials.Gemma, Sandra ; Campiani, Giuseppe ; Butini, Stefania ; B. P., Joshi; G., Kukreja; SANNA COCCONE, Salvatore; Bernetti, Matteo; M., Persico; Nacci, Vito; Fiorini, Isabella; E., Novellino; D., Taramelli; N., Basilico; S., Parapini; V., Yardley; S., Croft; S., KELLER MAERKI; M., Rottmann; R., Brun; M., Coletta; S., Marini; G., Guiso; S., Caccia; C., FattorussoNot applicable
142017Computational tool for fast in silico evaluation of hERG K+ channel affinityChemi, Giulia ; Gemma, Sandra ; Campiani, Giuseppe ; Brogi, Simone; Butini, Stefania ; Brindisi, Margherita Not applicable
152007Design and Synthesis of Potent Antimalarial Agents Based on Clotrimazole Scaffold: Exploring an Innovative Pharmacophore.Gemma, Sandra ; Campiani, Giuseppe ; Butini, Stefania ; B., Joshi; G., Kukreja; M., Persico; B., Catalanotti; E., Novellino; Fattorusso, E; Nacci, Vito; Savini, Luisa; D., Taramelli; N., Basilico; G., Morace; V., Yardley; C., FattorussoNot applicable
162008Design, synthesis, and structure-activity relationship studies of 4-quinolinyl- and 9-acrydinylhydrazones as potent antimalarial agents.C., Fattorusso; Campiani, Giuseppe ; G., Kukreja; M., Persico; Butini, Stefania ; Romano, MARIA PIA; Altarelli, Maria; S., Ros; Brindisi, Margherita ; Savini, Luisa; E., Novellino; Nacci, Vito; E., Fattorusso; S., Parapini; N., Basilico; D., Taramelli; V., Yardley; S., Croft; M., Borriello; Gemma, Sandra Not applicable
172016Development and Pharmacological Characterization of Selective Blockers of 2-Arachidonoyl Glycerol Degradation with Efficacy in Rodent Models of Multiple Sclerosis and PainBrindisi, Margherita ; Maramai, Samuele ; Gemma, Sandra ; Brogi, Simone; Grillo, Alessandro; Di Cesare Mannelli, Lorenzo; Gabellieri, Emanuele; Lamponi, Stefania ; Saponara, Simona; Gorelli, Beatrice; Tedesco, Daniele; Bonfiglio, Tommaso; Landry, Christophe; Jung, Kwang Mook; Armirotti, Andrea; Luongo, Livio; Ligresti, Alessia; Piscitelli, Fabiana; Bertucci, Carlo; Dehouck, Marie Pierre; Campiani, Giuseppe ; Maione, Sabatino; Ghelardini, Carla; Pittaluga, Anna; Piomelli, Daniele; Di Marzo, Vincenzo; Butini, Stefania Not applicable
182016Development of a practical and scalable route for the preparation of the deacetoxytubuvaline (dTuv) fragment of pretubulysin and analogsBrindisi, Margherita ; Samuele, Maramai; Alessandro, Grillo; Simone, Brogi; Butini, Stefania ; Ettore, Novellino; Campiani, Giuseppe ; Gemma, Sandra Not applicable
192009Development of Antitubercular Compounds Based on a 4-Quinolylhydrazone Scaffold. Further Structure-activity Relationship Studies.Gemma, Sandra ; Savini, Luisa; Altarelli, Maria; Tripaldi, Pierangela; Chiasserini, Luisa ; SANNA COCCONE, Salvatore; Vinod, Kumar; Camodeca, Caterina; Campiani, Giuseppe ; Ettore, Novellino; Sandra, Clarizio; Giovanni, Delogu; Butini, Stefania Not applicable
202005Development of molecular probes for the identification of extra interaction sites in the mid-gorge and peripheral sites of butyrylcholinesterase (BuChE). Rational design of novel, selective, and highly potent BuChE inhibitors.Campiani, Giuseppe ; Fattorusso, C; Butini, Stefania ; Gaeta, A; Agnusdei, M; Gemma, Sandra ; Persico, M; Catalanotti, B; Savini, Luisa; Nacci, Vito; Novellino, E; Holloway, Hw; Greig, Nh; Belinskaya, T; Fedorko, Jm; Saxena, A.Not applicable