| Issue Date | Title | Author(s) | Third Mission |
1 | 2011 | 1-Aryl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide: An effective scaffold for the design of either CB1 and CB2 receptor ligands | Piscitelli, F; Ligresti, A; LA REGINA, G; Gatti, V; Brizzi, Antonella ; Pasquini, Serena; Allarà, M; CARAI M. A., M; Novellino, E; Colombo, G; DI MARZO, V; Corelli, Federico ; Silvestri, R. | Not applicable |
2 | 2004 | 3D QSAR models of interactions between beta-tubulin and microtubule stabilizing antimitotic agents (MSAA): a survey on taxanes and epothilones | Manetti, Fabrizio ; L., Maccari; Corelli, Federico ; Botta, Maurizio | Not applicable |
3 | 2003 | 3D QSAR studies of the interaction between beta-tubulin and microtubule stabilizing antimitotic agents (MSAA). A combined pharmacophore generation and pseudoreceptor modeling approach applied to taxanes and epothilones | Botta, Maurizio ; Corelli, Federico ; S., Forli; L., Maccari; Manetti, Fabrizio | Not applicable |
4 | 2003 | 3D QSAR STUDIES OF THE INTERACTION BETWEEN BETA-TUBULIN AND MICROTUBULE STABILIZING ANTIMITOTIC AGENTS (MSAA). A PSEUDORECEPTOR MODEL FOR TAXANES BASED ON THE EXPERIMENTAL STRUCTURE OF TUBULIN. | L., Maccari; Corelli, Federico ; Manetti, Fabrizio ; Botta, Maurizio | Not applicable |
5 | 2009 | The 4-Quinolone-3-carboxylic Acid Motif as a Multivalent Scaffold in Medicinal Chemistry | Mugnaini, Claudia ; Pasquini, Serena; Corelli, Federico | Not applicable |
6 | 1993 | 5,6-Dihydro-5-[4-[4-(2-methoxyphenyl)-1- piperazinyl]butyl]-4H- pyrrolo[1,2-a][1,4]benzodiazepine-4,6-dione and Related Compounds as New 5-HT1A Receptor Ligands | Anzini, Maurizio ; Corelli, Federico ; A., Cagnotto; M., Skorupska | Not applicable |
7 | 2011 | Activation of the GABAB receptor prevents nicotine-induced locomotor stimulation in mice | Lobina, C.; Carai, M. A. M.; Froestl, W.; Mugnaini, Claudia ; Pasquini, Serena; Corelli, Federico ; G. e. s. s. a. G., L.; Colombo, G. | Not applicable |
8 | 2002 | Alpha1-Adrenoceptor Antagonists. 4. Pharmacophore-based Design, Synthesis, and Biological Evaluation of New Imidazo-, Benzimidazo-, and Indoloarylpiperazine Derivatives | L., Betti; Botta, Maurizio ; Corelli, Federico ; S., Corsano; M., Floridi; G., Giannaccini; L., Maccari; Manetti, Fabrizio ; G., Strappaghetti; Tafi, Andrea | Not applicable |
9 | 2003 | Alpha1-Adrenoceptor Antagonists. 6. Structural Optimization of Pyridazinone-Arylpiperazines. Study of the Influence on Affinity and Selectivity of Cyclic Substituents at the Pyridazinone Ring and Alkoxy Groups at the Arylpiperazine Moiety | L., Betti; Botta, Maurizio ; Corelli, Federico ; M., Floridi; G., Giannaccini; L., Maccari; Manetti, Fabrizio ; G., Strappaghetti | Not applicable |
10 | 2002 | alpha1-Adrenoceptor Antagonists. Rational Design, Synthesis and Biological Evaluation of New Trazodone-like Compounds | L., Betti; Botta, Maurizio ; Corelli, Federico ; M., Floridi; P., Fossa; G., Giannaccini; Manetti, Fabrizio ; G., Strappaghetti; S., Corsano | Not applicable |
11 | 2019 | Anti-addictive properties of COR659 – Additional pharmacological evidence and comparison with a series of novel analogues | Maccioni, Paola; Colombo, Giancarlo; Lorrai, Irene; Fara, Federica; Carai, Mauro A. M.; Gessa, Gian Luigi; Brizzi, Antonella ; Mugnaini, Claudia ; Corelli, Federico | Not applicable |
12 | 2002 | Antifungal agents. 10. New derivatives of 1-[(Aryl)[4-aryl-1H-pyrrol-3-yl]methyl]-1H-imidazole, synthesis, anti-Candida activity and Quantitative Structure-Analysis Relationship studies | Tafi, Andrea ; R., Costi; Botta, Maurizio ; R., DI SANTO; Corelli, Federico ; Massa, Silvio; A., Ciacci; Manetti, Fabrizio ; M., Artico | Not applicable |
13 | 2005 | Antifungal Agents. 11.N-Substituted Derivatives of 1-[(Aryl)(4-aryl-1H-pyrrol-3yl)methyl]-1H-imidazole: Synthesis, Anti-Candida Activity, and QSAR Studies | Di Santo, Roberto; Tafi, Andrea ; Costi, Roberta; Botta, Maurizio ; Artico, Marino; Corelli, Federico ; Forte, Michela; Caporuscio, Fabiana; Angiolella, Letizia; Palamara, Anna Teresa | Not applicable |
14 | 2015 | Anxiety-like behaviors at the end of the nocturnal period in sP rats with a “history” of unpredictable, limited access to alcohol. | Colombo, G.; Lobina, C.; Maccioni, P.; Carai, M. A. M.; Lorrai, I.; Zaru, A.; Contini, A.; Mugnaini, Claudia ; Corelli, Federico ; Gessa, G. | Not applicable |
15 | 2002 | Arylpiperazines with high affinity toward a1-adrenergic receptors | Manetti, Fabrizio ; Corelli, Federico ; Strappaghetti, G; Botta, Maurizio | Not applicable |
16 | 2012 | The bioisosteric concept applied to cannabinoid ligands | Mugnaini, Claudia ; Pasquini, Serena; Corelli, Federico | Not applicable |
17 | 2000 | Builiding a pharmacophore model for a novel class of antitubercular compounds. | Manetti, Fabrizio ; Corelli, Federico ; Biava, M; Fioravanti, R; Porretta, Gc; Botta, Maurizio | Not applicable |
18 | 1996 | Characterization and Differentiation of Heterocyclic Isomers. Part 2. Mass Spectrometry and Molecular Orbital Calculations on Pyrrolo[1,2-a][1,4]benzodiazepin-4-one, -6-one, -4,6-dione | Giorgi, Gianluca ; Anzini, Maurizio ; Cappelli, Andrea ; Corelli, Federico ; Vomero, Salvatore | Not applicable |
19 | 2012 | Characterization of COR627 and COR628, two novel positive allosteric modulators of the GABA B receptor | Castelli, M. P.; Casu, A.; Casti, P.; Lobina, C.; Carai, M. A. M.; Colombo, G.; Solinas, M.; Giunta, D.; Mugnaini, Claudia ; Pasquini, Serena; Tafi, Andrea ; Brogi, Simone; Gessa, G. L.; Corelli, Federico | Not applicable |
20 | 1999 | Chiral Azole Derivatives, 3. Synthesis of the Enantiomers of the Potent Aromatase Inhibitor 1-[2-Benzofuranyl(4-chlorophenyl)methyl]-1H-imidazole | Messina, F.; Botta, Maurizio ; Corelli, Federico ; Mugnaini, Claudia | Not applicable |