Full Name
Botta, Maurizio
 
DBCF community
 
Discipline (SSD)
CHIM/08 - Chimica Farmaceutica
 
Email UNISI
maurizio.botta@unisi.it
 
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Publications
(Articles)

Results 1-20 of 387 (Search time: 0.002 seconds).

Issue DateTitleAuthor(s)Third Mission
120091,5-Diaryl-2-ethyl pyrrole derivatives as antimycobacterial agents: design, synthesis, and microbiological evaluationM., Biava; G. C., Porretta; G., Poce; A., DE LOGU; R., Meleddu; E., DE ROSSI; Manetti, Fabrizio ; Botta, Maurizio Not applicable
220051,5-Diarylpyrrole-3-acetic Acids and Esters as Novel Classes of Potent and Highly Selective Cyclooxygenase-2 InhibitorsBiava, M.; Porretta, G. C.; Cappelli, Andrea ; Vomero, S.; Manetti, Fabrizio ; Botta, Maurizio ; Sautebin, L.; Rossi, A.; Makovec, F.; Anzini, Maurizio Not applicable
320081,5-Diphenylpyrrole Derivatives as Antimycobacterial Agents. Probing the Influence on Antimycobacterial Activity of Lipophilic Substituents at the Phenyl RingsBiava, M; PORRETTA G., C; Poce, G; DE LOGU, A; Saddi, M; Meleddu, R; Manetti, Fabrizio ; DE ROSSI, E; Botta, Maurizio Not applicable
420081-[(3-Aryloxy-3-aryl)propyl]-2H-imidazoles, new imidazoles with potent activity against Candida albicans and dermatophytes. Synthesis, structure-activity relationship, and molecular modeling studiesG., LA REGINA; F., D'Auria; Tafi, Andrea ; F., Piscitelli; S., Olla; F., Caporuscio; L., Nencioni; R., Cirilli; F., LA TORRE; N., RODRIGUES DE MELO; S., Kelly; D., Lamb; M., Artico; Botta, Maurizio ; A., Palamara; R., SilvestriNot applicable
520142-Aminothiazolones as anti-hiv agents that act as gp120-cd4 inhibitorsTiberi, Marika; Tintori, Cristina; Ceresola, Elisa Rita; Fazi, Roberta; Zamperini, Claudio; Calandro, Pierpaolo; Franchi, Luigi; Selvaraj, Manikandan; Botta, Lorenzo; Sampaolo, Michela; Saita, Diego; Ferrarese, Roberto; Clementi, Massimo; Canducci, Filippo; Botta, Maurizio Not applicable
620102-Hydroxypropyl-β-cyclodextrin strongly improves water solubility and anti-proliferative activity of pyrazolo[3,4-d]pyrimidines Src-Abl dual inhibitors.Dreassi, Elena ; Zizzari, ALESSANDRA TANIA; Mori, Mattia ; Filippi, Irene; Belfiore, Amalia; Naldini, Antonella; Carraro, Fabio; Santucci, Annalisa ; Schenone, S; Botta, Maurizio Not applicable
720163-Arylidene-N-hydroxyoxindoles: A New Class of Compounds Endowed with Antitumor ActivityMusso, Loana; Cincinelli, Raffaella; Zuco, Valentina; Decesare, Michelandrea; Zunino, Franco; Fallacara, Anna Lucia; Botta, Maurizio ; Dallavalle, SabrinaNot applicable
820093D QSAR models built on structure-based alignments of Abl tyrosine kinase inhibitors.Falchi, F; Manetti, Fabrizio ; Carraro, Fabio; Naldini, Antonella; Maga, G; Crespan, E; Schenone, S; Bruno, O; Brullo, C; Botta, Maurizio Not applicable
920043D QSAR models of interactions between beta-tubulin and microtubule stabilizing antimitotic agents (MSAA): a survey on taxanes and epothilonesManetti, Fabrizio ; L., Maccari; Corelli, Federico ; Botta, Maurizio Not applicable
1020033D QSAR studies of the interaction between beta-tubulin and microtubule stabilizing antimitotic agents (MSAA). A combined pharmacophore generation and pseudoreceptor modeling approach applied to taxanes and epothilonesBotta, Maurizio ; Corelli, Federico ; S., Forli; L., Maccari; Manetti, Fabrizio Not applicable
1120033D QSAR STUDIES OF THE INTERACTION BETWEEN BETA-TUBULIN AND MICROTUBULE STABILIZING ANTIMITOTIC AGENTS (MSAA). A PSEUDORECEPTOR MODEL FOR TAXANES BASED ON THE EXPERIMENTAL STRUCTURE OF TUBULIN.L., Maccari; Corelli, Federico ; Manetti, Fabrizio ; Botta, Maurizio Not applicable
1220164,6-Diphenylpyridines as Promising Novel Anti-Influenza Agents Targeting the PA-PB1 Protein-Protein Interaction: Structure-Activity Relationships Exploration with the Aid of Molecular ModelingTrist, Iuni M. L.; Nannetti, Giulio; Tintori, Cristina; Fallacara, ANNA LUCIA; Deodato, Davide; Mercorelli, Beatrice; Palù, Giorgio; Wijtmans, Maikel; Gospodova, Tzveta; Edink, Ewald; Verheij, Mark; De Esch, Iwan; Viteva, Lilia; Loregian, Arianna; Botta, Maurizio Not applicable
1320094­-Amino­substituted pyrazolo[3,4­d]pyrimidines: synthesis and biological propertiesS., Schenone; O., Bruno; Radi, Marco; Botta, Maurizio Not applicable
1420205,6-Dihydroxypyrimidine Scaffold to Target HIV-1 Nucleocapsid ProteinMalancona, Savina; Mori, Mattia ; Fezzardi, Paola; Santoriello, Marisabella; Basta, Andreina; Nibbio, Martina; Kovalenko, Lesia; Speziale, Roberto; Battista, Maria Rosaria; Cellucci, Antonella; Gennari, Nadia; Monteagudo, Edith; Di Marco, Annalise; Giannini, Alessia; Sharma, Rajhans; Pires, Manuel; Real, Eleonore; Zazzi, Maurizio; Dasso Lang, Maria Chiara; De Forni, Davide; Saladini, Francesco; Mely, Yves; Summa, Vincenzo; Harper, Steven; Botta, Maurizio Not applicable
1519905-HT and Benzodiazepine Receptor Ligands. III. Synthesis and Receptor Affinities of 1,2,4,-Triazolo[4',3':1,6]pyridazino[4,5-b]quinoline and 2,3-Dihydro-9-phenyl-1H-pyrrolo[3,4-b]quinoline-1-one DerivativesAnzini, Maurizio ; Cappelli, Andrea ; Vomero, Salvatore; Botta, Maurizio ; A., CagnottoNot applicable
162010A1 receptors ligands: past, present and future trendsS., Schenone; C., Brullo; F., Musumeci; O., Bruno; Botta, Maurizio Not applicable
172018Alkyl-guanidine Compounds as Potent Broad-Spectrum Antibacterial Agents: Chemical Library Extension and Biological CharacterizationPasero, Carolina; D'Agostino, Ilaria ; De Luca, Filomena; Zamperini, Claudio; Deodato, Davide; Truglio, Giuseppina Ivana ; Sannio, Filomena; Del Prete, Rosita; Ferraro, Teresa; Visaggio, Daniela; Mancini, Arianna ; Guglielmi, Mario B.; Visca, Paolo; Docquier, Jean-Denis; Botta, Maurizio Not applicable
182009Alkyne-enol ether cross-metathesis in the presence of CuSO. Direct formation of 3-substituted crotonaldehydes in aqueous mediumCastagnolo, Daniele; Botta, Lorenzo; Botta, Maurizio Not applicable
192013Allosteric Inhibitors of Bcr-Abl: Towards Novel Myristate-Pocket Binders.Botta, Maurizio ; Schenone, S.; Botta, Maurizio Not applicable
202002Alpha1-Adrenoceptor Antagonists. 4. Pharmacophore-based Design, Synthesis, and Biological Evaluation of New Imidazo-, Benzimidazo-, and Indoloarylpiperazine DerivativesL., Betti; Botta, Maurizio ; Corelli, Federico ; S., Corsano; M., Floridi; G., Giannaccini; L., Maccari; Manetti, Fabrizio ; G., Strappaghetti; Tafi, Andrea Not applicable