Mori, Mattia
Personal picture

Full Name
Mori, Mattia
DBCF community
Discipline (SSD)
CHIM/08 - Chimica Farmaceutica
Email UNISI
mattia.mori@unisi.it
ORCID





ERC sector
PE5_18
Publications
(Articles)
Results 1-20 of 88 (Search time: 0.005 seconds).
Issue Date | Title | Author(s) | Third Mission | |
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1 | 2020 | 14-3-3 binding creates a memory of kinase action by stabilizing the modified state of phospholamban | Menzel, J.; Kownatzki-Danger, D.; Tokar, S.; Ballone, A.; Unthan-Fechner, K.; Kilisch, M.; Lenz, C.; Urlaub, H.; Mori, Mattia ; Ottmann, C.; Shattock, M. J.; Lehnart, S. E.; Schwappach, B. | Not applicable |
2 | 2019 | 1H-NMR metabolomics reveals the Glabrescione B exacerbation of glycolytic metabolism beside the cell growth inhibitory effect in glioma | D'Alessandro, G.; Quaglio, D.; Monaco, L.; Lauro, C.; Ghirga, F.; Ingallina, C.; De Martino, M.; Fucile, S.; Porzia, A.; Di Castro, M. A.; Bellato, F.; Mastrotto, F.; Mori, Mattia ; Infante, P.; Turano, P.; Salmaso, S.; Caliceti, P.; Di Marcotullio, L.; Botta, B.; Ghini, V.; Limatola, C. | Not applicable |
3 | 2010 | 2-Hydroxypropyl-β-cyclodextrin strongly improves water solubility and anti-proliferative activity of pyrazolo[3,4-d]pyrimidines Src-Abl dual inhibitors. | Dreassi, Elena ; Zizzari, ALESSANDRA TANIA; Mori, Mattia ; Filippi, Irene; Belfiore, Amalia; Naldini, Antonella; Carraro, Fabio; Santucci, Annalisa ; Schenone, S; Botta, Maurizio | Not applicable |
4 | 2020 | 5,6-Dihydroxypyrimidine Scaffold to Target HIV-1 Nucleocapsid Protein | Malancona, Savina; Mori, Mattia ; Fezzardi, Paola; Santoriello, Marisabella; Basta, Andreina; Nibbio, Martina; Kovalenko, Lesia; Speziale, Roberto; Battista, Maria Rosaria; Cellucci, Antonella; Gennari, Nadia; Monteagudo, Edith; Di Marco, Annalise; Giannini, Alessia; Sharma, Rajhans; Pires, Manuel; Real, Eleonore; Zazzi, Maurizio; Dasso Lang, Maria Chiara; De Forni, Davide; Saladini, Francesco; Mely, Yves; Summa, Vincenzo; Harper, Steven; Botta, Maurizio | Not applicable |
5 | 2020 | Alvaxanthone, a thymidylate synthase inhibitor with nematocidal and tumoricidal activities | Maj, P.; Mori, Mattia ; Sobich, J.; Markowicz, J.; Uram, L.; Zielinski, Z.; Quaglio, D.; Calcaterra, A.; Cau, Y.; Botta, B.; Rode, W. | Not applicable |
6 | 2020 | A chalcone derivative binds a putative allosteric site of YopH: Inhibition of a virulence factor of Yersinia | de Souza, A. C. A.; Mori, Mattia ; Sens, L.; Rocha, R. F.; Tizziani, T.; de Souza, L. F. S.; Domeneghini Chiaradia-Delatorre, L.; Botta, Maurizio ; Nunes, R. J.; Terenzi, H.; Menegatti, A. C. O. | Not applicable |
7 | 2019 | Chalcones and Chalcone-mimetic Derivatives as Notch Inhibitors in a Model of T-cell Acute Lymphoblastic Leukemia | Quaglio, D.; Zhdanovskaya, N.; Tobajas, G.; Cuartas, V.; Balducci, S.; Christodoulou, M. S.; Fabrizi, G.; Gargantilla, M.; Priego, E. -M.; Carmona Pestania, A.; Passarella, D.; Screpanti, I.; Botta, B.; Palermo, R.; Mori, Mattia ; Ghirga, F.; Perez-Perez, M. -J. | Not applicable |
8 | 2019 | Chemically stable inhibitors of 14-3-3 protein–protein interactions derived from BV02 | Iralde-Lorente, Leire; Cau, Ylenia; Clementi, Letizia; Franci, Lorenzo; Tassone, Giusy ; Valensin, Daniela ; Mori, Mattia ; Angelucci, Adriano; Chiariello, Mario; Botta, Maurizio | Not applicable |
9 | 2020 | A Class of Potent Inhibitors of the HIV-1 Nucleocapsid Protein Based on Aminopyrrolic Scaffolds | Ciaco, S.; Humbert, N.; Real, E.; Boudier, C.; Francesconi, O.; Roelens, S.; Nativi, C.; Seguin-Devaux, C.; Mori, Mattia ; Mely, Y. | Not applicable |
10 | 2015 | Click reaction as a tool to combine pharmacophores: The case of Vismodegib | Christodoulou, Michael S; Mori, Mattia ; Pantano, Rebecca; Alfonsi, Romina; Infante, Paola; Botta, Maurizio ; Damia, Giovanna; Ricci, Francesca; Sotiropoulou, Panagiota A.; Liekens, Sandra; Botta, Bruno; Passarella, Daniele | Not applicable |
11 | 2013 | A combination strategy to inhibit Pim-1: synergism between noncompetitive and ATP-competitive inhibitors | Mori, Mattia ; Tintori, Cristina; Christopher, R. S. A.; Radi, M.; Schenone, S.; Musumeci, F.; Brullo, C.; Sanità, P.; Delle Monache, S.; Angelucci, A.; Kissova, M.; Crespan, E.; Maga, G.; Botta, Maurizio | Not applicable |
12 | 2011 | Computational techniques are valuable tools for the identification of protein-protein interaction inhibitors: the 14-3-3σ case | Corradi, V; Mancini, M; Santucci, Ma; Carlomagno, T; Sanfelice, D; Mori, Mattia ; Vignaroli, G; Falchi, F; Manetti, Fabrizio ; Radi, M; Botta, Maurizio | Not applicable |
13 | 2018 | Current trends in Hedgehog signaling pathway inhibition by small molecules | Ghirga, F.; Mori, Mattia ; Infante, P. | Not applicable |
14 | 2018 | Design, synthesis, SAR and biological investigation of 3-(carboxymethyl)rhodanine and aminothiazole inhibitors of Mycobacterium tuberculosis Zmp1 | Mori, Mattia ; Deodato, Davide; Kasula, Mohan; Ferraris, Davide M.; Sanna, Adriana; De Logu, Alessandro; Rizzi, Menico; Botta, Maurizio | Not applicable |
15 | 2017 | Differentially activated Src kinase in chemo-naive human primary osteosarcoma cells and effects of a Src kinase inhibitor | Laschi, Marcella; Bernardini, Giulia ; Geminiani, Michela ; Manetti, Fabrizio ; Mori, Mattia ; Spreafico, Adriano; Campanacci, Domenico; Capanna, Rodolfo; Schenone, Silvia; Botta, Maurizio ; Santucci, Annalisa | Not applicable |
16 | 2014 | Discovery of 14-3-3 Protein-Protein Interaction Inhibitors that Sensitize Multidrug-Resistant Cancer Cells to Doxorubicin and the Akt Inhibitor GSK690693 | Mori, Mattia ; Vignaroli, Giulia; Cau, Ylenia; Dinić, J; Hill, R; Rossi, M; Colecchia, D; Pešić, M; Link, W; Chiariello, M; Ottmann, C; Botta, Maurizio | Not applicable |
17 | 2013 | Discovery of a New Class of Potent MMP Inhibitors by Structure-Based Optimization of the Arylsulfonamide Scaffold | Mori, Mattia ; Massaro, Assunta; Calderone, Vito; Fragai, Marco; Luchinat, Claudio; Mordini, Alessandro | Not applicable |
18 | 2016 | Discovery of in vitro antitubercular agents through in silico ligand-based approaches | De Vita, Daniela; Pandolfi, Fabiana; Cirilli, Roberto; SCIPIONE, LUIGI; Di Santo, Roberto; Friggeri, Laura; Mori, Mattia ; FIORUCCI, DIEGO; Maccari, Giorgio; Christopher, Robert Selwyne Arul; ZAMPERINI, CLAUDIO; Pau, Valentina; De Logu, Alessandro; Tortorella, Silvano; Botta, Maurizio | Not applicable |
19 | 2013 | Discovery of Mycobacterium tuberculosis protein tyrosine phosphatase B (PtpB) inhibitors from natural products | Mascarello, A; Mori, Mattia ; Chiaradia Delatorre, Ld; Menegatti, Ac; Delle Monache, F; Ferrari, F; Yunes, Ra; Nunes, Rj; Terenzi, H; Botta, B; Botta, Maurizio | Not applicable |
20 | 2020 | Discovery of small molecule inhibitors of Leishmania braziliensis Hsp90 chaperone | Batista, F. A. H.; Ramos, S. L.; Tassone, Giusy ; Leitao, A.; Montanari, C. A.; Botta, Maurizio ; Mori, Mattia ; Borges, J. C. | Not applicable |