Manetti, Fabrizio
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Full Name
Manetti, Fabrizio
DBCF community
Discipline (SSD)
CHIM/08 - Chimica Farmaceutica
Email UNISI
fabrizio.manetti@unisi.it





Publications
(Articles)
Results 1-20 of 160 (Search time: 0.009 seconds).
Issue Date | Title | Author(s) | Third Mission | |
---|---|---|---|---|
1 | 2009 | 1,5-Diaryl-2-ethyl pyrrole derivatives as antimycobacterial agents: design, synthesis, and microbiological evaluation | M., Biava; G. C., Porretta; G., Poce; A., DE LOGU; R., Meleddu; E., DE ROSSI; Manetti, Fabrizio ; Botta, Maurizio | Not applicable |
2 | 2005 | 1,5-Diarylpyrrole-3-acetic Acids and Esters as Novel Classes of Potent and Highly Selective Cyclooxygenase-2 Inhibitors | Biava, M.; Porretta, G. C.; Cappelli, Andrea ; Vomero, S.; Manetti, Fabrizio ; Botta, Maurizio ; Sautebin, L.; Rossi, A.; Makovec, F.; Anzini, Maurizio | Not applicable |
3 | 2008 | 1,5-Diphenylpyrrole Derivatives as Antimycobacterial Agents. Probing the Influence on Antimycobacterial Activity of Lipophilic Substituents at the Phenyl Rings | Biava, M; PORRETTA G., C; Poce, G; DE LOGU, A; Saddi, M; Meleddu, R; Manetti, Fabrizio ; DE ROSSI, E; Botta, Maurizio | Not applicable |
4 | 2002 | 2-Substituted 5-Acetyl-1,6-Dihydro-6-oxo-3-pyridinecarboxylates: Synthesis and Cardiotonic Activity | P., Dorigo; M., Floreani; P., Fossa; Manetti, Fabrizio ; G., Menozzi; L., Mosti | Not applicable |
5 | 2009 | 3D QSAR models built on structure-based alignments of Abl tyrosine kinase inhibitors. | Falchi, F; Manetti, Fabrizio ; Carraro, Fabio; Naldini, Antonella; Maga, G; Crespan, E; Schenone, S; Bruno, O; Brullo, C; Botta, Maurizio | Not applicable |
6 | 2004 | 3D QSAR models of interactions between beta-tubulin and microtubule stabilizing antimitotic agents (MSAA): a survey on taxanes and epothilones | Manetti, Fabrizio ; L., Maccari; Corelli, Federico ; Botta, Maurizio | Not applicable |
7 | 2003 | 3D QSAR studies of the interaction between beta-tubulin and microtubule stabilizing antimitotic agents (MSAA). A combined pharmacophore generation and pseudoreceptor modeling approach applied to taxanes and epothilones | Botta, Maurizio ; Corelli, Federico ; S., Forli; L., Maccari; Manetti, Fabrizio | Not applicable |
8 | 2003 | 3D QSAR STUDIES OF THE INTERACTION BETWEEN BETA-TUBULIN AND MICROTUBULE STABILIZING ANTIMITOTIC AGENTS (MSAA). A PSEUDORECEPTOR MODEL FOR TAXANES BASED ON THE EXPERIMENTAL STRUCTURE OF TUBULIN. | L., Maccari; Corelli, Federico ; Manetti, Fabrizio ; Botta, Maurizio | Not applicable |
9 | 2017 | 4-Hydroxyphenylpyruvate Dioxygenase and Its Inhibition in Plants and Animals: Small Molecules as Herbicides and Agents for the Treatment of Human Inherited Diseases | Santucci, Annalisa ; Bernardini, Giulia ; Braconi, Daniela ; Petricci, Elena ; Manetti, Fabrizio | Not applicable |
10 | 2012 | Acylthiourea, Acylurea and Acylguanidine Derivatives with potent Hedgehog inhibiting Activity | Solinas, A; Faure, H; Roudaut, H; Traiffort, E; Schoenfelder, A; Mann, A; Manetti, Fabrizio ; Taddei, Maurizio ; Ruat, M. | Not applicable |
11 | 2002 | Alpha1-Adrenoceptor Antagonists. 4. Pharmacophore-based Design, Synthesis, and Biological Evaluation of New Imidazo-, Benzimidazo-, and Indoloarylpiperazine Derivatives | L., Betti; Botta, Maurizio ; Corelli, Federico ; S., Corsano; M., Floridi; G., Giannaccini; L., Maccari; Manetti, Fabrizio ; G., Strappaghetti; Tafi, Andrea | Not applicable |
12 | 2003 | Alpha1-Adrenoceptor Antagonists. 6. Structural Optimization of Pyridazinone-Arylpiperazines. Study of the Influence on Affinity and Selectivity of Cyclic Substituents at the Pyridazinone Ring and Alkoxy Groups at the Arylpiperazine Moiety | L., Betti; Botta, Maurizio ; Corelli, Federico ; M., Floridi; G., Giannaccini; L., Maccari; Manetti, Fabrizio ; G., Strappaghetti | Not applicable |
13 | 2002 | alpha1-Adrenoceptor Antagonists. Rational Design, Synthesis and Biological Evaluation of New Trazodone-like Compounds | L., Betti; Botta, Maurizio ; Corelli, Federico ; M., Floridi; P., Fossa; G., Giannaccini; Manetti, Fabrizio ; G., Strappaghetti; S., Corsano | Not applicable |
14 | 2005 | The anti-HIV activity of ADS-J1 targets the HIV-1 gp120 | ARMAND UGON, M.; CLOTET CODINA, I.; Tintori, Cristina; Manetti, Fabrizio ; Clotet, B.; Botta, Maurizio ; Este, J. A. | Not applicable |
15 | 2002 | Antifungal agents. 10. New derivatives of 1-[(Aryl)[4-aryl-1H-pyrrol-3-yl]methyl]-1H-imidazole, synthesis, anti-Candida activity and Quantitative Structure-Analysis Relationship studies | Tafi, Andrea ; R., Costi; Botta, Maurizio ; R., DI SANTO; Corelli, Federico ; Massa, Silvio; A., Ciacci; Manetti, Fabrizio ; M., Artico | Not applicable |
16 | 2006 | Antimycobacterial Agents. Novel Diarylpyrrole Derivatives of BM212 Endowed with High Activity toward Mycobacterium tuberculosis and Low Cytotoxicity | M., Biava; G. C., Porretta; G., Poce; S., Supino; D., Deidda; R., Pompei; P., Molicotti; Manetti, Fabrizio ; Botta, Maurizio | Not applicable |
17 | 2004 | Antimycobacterial compounds. New pyrrole derivatives of BM212 | Biava, M.; Porretta, G. C.; Deidda, D.; Pompei, R.; Tafi, Andrea ; Manetti, Fabrizio | Not applicable |
18 | 2005 | Antimycobacterial compounds. Optimization of the BM212 structure, the lead compound for a new pyrrole derivative class | Biava, M; Porretta, Gc; Poce, G; Deidda, D; Pompei, R; Tafi, Andrea ; Manetti, Fabrizio | Not applicable |
19 | 2004 | Antiproliferative activity of new 1-aryl-4-amino-1H-pyrazolo[3,4-d]pyrimidine derivatives toward the human epidermoid carcinoma A431 cell line. | Schenone, S.; Bruno, O.; Bondavalli, F.; Ranise, A.; Mosti, L.; Menozzi, G.; Fossa, P.; Donnini, Sandra; Santoro, A.; Ziche, Marina; Manetti, Fabrizio ; Botta, Maurizio | Not applicable |
20 | 2008 | Antiproliferative and proapoptotic activities of new pyrazolo[3,4-d]pyrimidine derivative Src kinase inhibitors in human osteosarcoma cells. | Spreafico, A; Schenone, S; Serchi, T; Orlandini, Maurizio ; Angelucci, A; Magrini, D; Bernardini, Giulia ; Collodel, Giulia; DI STEFANO, Anna; Tintori, C; Bologna, M; Manetti, Fabrizio ; Botta, Maurizio ; Santucci, Annalisa | Not applicable |