Browsing by Author Zamperini, Claudio
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Issue Date | Title | Author(s) | Third Mission |
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2014 | 2-Aminothiazolones as anti-hiv agents that act as gp120-cd4 inhibitors | Tiberi, Marika; Tintori, Cristina; Ceresola, Elisa Rita; Fazi, Roberta; Zamperini, Claudio; Calandro, Pierpaolo; Franchi, Luigi; Selvaraj, Manikandan; Botta, Lorenzo; Sampaolo, Michela; Saita, Diego; Ferrarese, Roberto; Clementi, Massimo; Canducci, Filippo; Botta, Maurizio | Not applicable |
2018 | Alkyl-guanidine Compounds as Potent Broad-Spectrum Antibacterial Agents: Chemical Library Extension and Biological Characterization | Pasero, Carolina; D'Agostino, Ilaria ; De Luca, Filomena; Zamperini, Claudio; Deodato, Davide; Truglio, Giuseppina Ivana ; Sannio, Filomena; Del Prete, Rosita; Ferraro, Teresa; Visaggio, Daniela; Mancini, Arianna ; Guglielmi, Mario B.; Visca, Paolo; Docquier, Jean-Denis; Botta, Maurizio | Not applicable |
2012 | A combined targeted/phenotypic approach for the identification of new antiangiogenics agents active on a zebrafish model:from in silico screening to cyclodextrin formulation | Botta, Maurizio ; Evensen, L.; Dreassi, Elena ; Zamperini, Claudio; Caporicci, M.; Falchi, Federico; Musumeci, A.; Schenone, S.; Lorens, J. B.; Botta, Maurizio | Not applicable |
2014 | Combining X-ray Crystallography and Molecular Modeling toward the Optimization of Pyrazolo[3,4-d]pyrimidines as Potent c-Src Inhibitors Active in Vivo against Neuroblastoma. | Tintori, Cristina; Fallacara, A. L.; Radi, Marco; Zamperini, Claudio; Dreassi, Elena ; Crespan, E.; Maga, G.; Schenone, S.; Musumeci, F.; Brullo, C.; Richters, A.; Gasparrini, F.; Angelucci, A.; Festuccia, C.; Delle Monache, S.; Rauh, D.; Botta, Maurizio | Not applicable |
2014 | CYP-dependent metabolism of antitumor pyrazolo[3,4-d]pyrimidine derivatives is characterized by an oxidative dechlorination reaction. | Zamperini, Claudio; Dreassi, Elena ; Vignaroli, Giulia; Botta, Maurizio ; Dragoni, S; Schenone, S; Musumeci, Francesca; Valoti, Massimo; Antiochia, R; Botta, Maurizio | Not applicable |
2019 | DDX3X Helicase Inhibitors as a New Strategy to Fight the West Nile Virus Infection | Brai, Annalaura; Martelli, Francesco; Riva, Valentina; Garbelli, Anna; Fazi, Roberta; Zamperini, Claudio; Pollutri, Alessandro; Falsitta, Lucia ; Ronzini, Stefania; Maccari, Laura; Maga, Giovanni; Giannecchini, Simone; Botta, Maurizio | Not applicable |
2020 | DDX3X inhibitors, an effective way to overcome HIV-1 resistance | Brai, Annalaura; Riva, Valentina; Saladini, Francesco; Zamperini, Claudio; Trivisani, Claudia Immacolata ; Garbelli, Anna; Pennisi, Carla; Giannini, Alessia; Boccuto, Adele; Bugli, Francesca; Martini, Maurizio; Sanguinetti, Maurizio; Dreassi, Elena ; Zazzi, Maurizio; Maga, Giovanni; Botta, Maurizio | Not applicable |
2013 | Design, synthesis, and biological evaluation of pyrazolo[3,4-d]pyrimidines active in vivo on the Bcr-Abl T315I mutant | Botta, Maurizio ; Tintori, Cristina; Musumeci, F.; Brullo, C.; Zamperini, Claudio; Dreassi, Elena ; Fallacara, ANNA LUCIA; Vignaroli, Giulia; Crespan, E.; Zanoli, S.; Laurenzana, Ilaria; Filippi, I.; Maga, G.; Schenone, S.; Angelucci, A.; Botta, Maurizio | Not applicable |
2011 | Design, synthesis, biological activity and ADME properties of pyrazolo[3,4-d]pyrimidines active in hypoxic human leukemia cells: a lead optimization study | Radi, Marco; Dreassi, Elena ; C., Brullo; E., Crespan; Tintori, Cristina; V., Bernardo; Valoti, Massimo; Zamperini, Claudio; H., Daigl; F., Musumeci; Carraro, Fabio; Naldini, Antonella; Filippi, Irene; G., Maga; S., Schenone; Botta, Maurizio | Not applicable |
2016 | Development and in Vitro Evaluation of a Microbicide Gel Formulation for a Novel Non-Nucleoside Reverse Transcriptase Inhibitor Belonging to the N-Dihydroalkyloxybenzyloxopyrimidines (N-DABOs) Family | Tintori, Cristina; Brai, Annalaura; DASSO LANG, MARIA CHIARA; Deodato, Davide; Greco, Antonia Michela; Bizzarri, Bruno Mattia; Cascone, Lorena; Casian, Alexandru; Zamperini, Claudio; Dreassi, Elena ; Crespan, Emmanuele; Maga, Giovanni; Vanham, Guido; Ceresola, Elisa; Canducci, Filippo; Ariën, Kevin K.; Botta, Maurizio | Not applicable |
2018 | Efficient optimization of pyrazolo[3,4-d]pyrimidines derivatives as c-Src kinase inhibitors in neuroblastoma treatment | Molinari, Alessio; Fallacara, Anna Lucia; Di Maria, Salvatore ; Zamperini, Claudio; Poggialini, Federica ; Musumeci, Francesca; Schenone, Silvia; Angelucci, Adriano; Colapietro, Alessandro; Crespan, Emmanuele; Kissova, Miroslava; Maga, Giovanni; Botta, Maurizio | Not applicable |
2011 | Identification of potent c-Src inhibitors strongly affecting the proliferation of human neuroblastoma cells. | Botta, Maurizio ; Brullo, C.; Crespan, E.; Tintori, Cristina; Musumeci, F.; Biava, M.; Schenone, S.; Dreassi, Elena ; Zamperini, Claudio; Maga, G.; Pagano, D.; Angelucci, A.; Bologna, M.; Botta, Maurizio | Not applicable |
2016 | Improvement of pyrazolo[3,4-d]pyrimidines pharmacokinetic properties: Nanosystem approaches for drug delivery | Vignaroli, Giulia; Calandro, Pierpaolo; Zamperini, Claudio; Coniglio, Federica; Iovenitti, Giulia ; Tavanti, Matteo; Colecchia, David; Dreassi, Elena ; Valoti, Massimo; Schenone, Silvia; Chiariello, Mario; Botta, Maurizio | Not applicable |
2014 | Indolylarylsulfones carrying a heterocyclic tail as very potent and broad spectrum HIV-1 non-nucleoside reverse transcriptase inhibitors | Famiglini, V.; La Regina, G.; Coluccia, A.; Pelliccia, S.; Brancale, A.; Maga, G.; Crespan, E.; Badia, R.; Riveira Muñoz, E.; Esté, J. A.; Ferretti, R.; Cirilli, R.; Zamperini, Claudio; Botta, Maurizio ; Schols, D.; Limongelli, V.; Agostino, B.; Novellino, E.; Silvestri, R. | Not applicable |
2015 | New 1-phenyl-5-(1 H -pyrrol-1-yl)-1 H -pyrazole-3-carboxamides inhibit hepatitis C virus replication via suppression of cyclooxygenase-2 | Manvar, Dinesh; Pelliccia, Sveva; La Regina, Giuseppe; Famiglini, Valeria; Coluccia, Antonio; Ruggieri, Anna; Anticoli, Simona; Lee, Jin Ching; Basu, Amartya; Cevik, Ozge; Nencioni, Lucia; Palamara, Anna Teresa; Zamperini, Claudio; Botta, Maurizio ; Neyts, Johan; Leyssen, Pieter; Kaushik Basu, Neerja; Silvestri, Romano | Not applicable |
2014 | New Pyrazolobenzothiazine Derivatives as Hepatitis C Virus NS5B Polymerase Palm Site I Inhibitors | Giuseppe, Manfroni; Dinesh, Manvar; Maria, Letizia Barreca; Neerja, Kaushik Basu; Pieter, Leyssen; Jan, Paeshuyse; Rolando, Cannalire; Nunzio, Iraci; Amartya, Basu; Maxim, Chudaev; Zamperini, Claudio; Dreassi, Elena ; Stefano, Sabatini; Oriana, Tabarrini; Johan, Neyts; Violetta, Cecchetti | Not applicable |
2019 | A New Strategy for Glioblastoma Treatment: In Vitro and In Vivo Preclinical Characterization of Si306, a Pyrazolo[3,4-d]Pyrimidine Dual Src/P-Glycoprotein Inhibitor | Fallacara, Anna Lucia; Zamperini, Claudio; Podolski-Renić, Ana; Dinić, Jelena; Stanković, Tijana; Stepanović, Marija; Mancini, Arianna ; Rango, Enrico ; Iovenitti, Giulia ; Molinari, Alessio; Bugli, Francesca; Sanguinetti, Maurizio; Torelli, Riccardo; Martini, Maurizio; Maccari, Laura; Valoti, Massimo; Dreassi, Elena ; Botta, Maurizio ; Pešić, Milica; Schenone, Silvia | Not applicable |
2018 | Plasmin-Binding Tripeptide-Decorated Liposomes Loading Pyrazolo[3,4- d]pyrimidines for Targeting Hepatocellular Carcinoma | Calandro, Pierpaolo; Iovenitti, Giulia ; Zamperini, Claudio; Candita, Francesca; Dreassi, Elena ; Chiariello, Mario; Angelucci, Adriano; Schenone, Silvia; Botta, Maurizio ; Mancini, Arianna | Not applicable |
2019 | Presence of Destruxin A and Beauvericin in cereals | Dreassi, Elena ; Zamperini, Claudio; Cito, Annarita; Francardi, Valeria; Botta, Maurizio | Not applicable |
2017 | Prodrugs of pyrazolo[3,4-d]pyrimidines: from library synthesis to evaluation as potential anticancer agents in an orthotopic glioblastoma model | Vignaroli, Giulia; Iovenitti, Giulia ; Zamperini, Claudio; Coniglio, Federica; Calandro, Pierpaolo; Molinari, Alessio; Fallacara, ANNA LUCIA; Sartucci, Andrea; Calgani, Alessia; Colecchia, David; Mancini, Andrea; Festuccia, Claudio; Dreassi, Elena ; Valoti, Massimo; Musumeci, Francesca; Chiariello, Mario; Angelucci, Adriano; Botta, Maurizio ; Schenone, Silvia | Not applicable |