Browsing by Author Radi, Marco

Showing results 1 to 20 of 20
Issue DateTitleAuthor(s)Third Mission
20094­-Amino­substituted pyrazolo[3,4­d]pyrimidines: synthesis and biological propertiesS., Schenone; O., Bruno; Radi, Marco; Botta, Maurizio Not applicable
2010Arylation of 2-Furyl 4-Fluorophenyl Ketone: an extension of Heck Chemistry towards Novel Integrase InhibitorsFranchi, Luigi; Rinaldi, Marta; Vignaroli, Giulia; Innitzer, Anna; Radi, Marco; Botta, Maurizio Not applicable
2014Combining X-ray Crystallography and Molecular Modeling toward the Optimization of Pyrazolo[3,4-d]pyrimidines as Potent c-Src Inhibitors Active in Vivo against Neuroblastoma.Tintori, Cristina; Fallacara, A. L.; Radi, Marco; Zamperini, Claudio; Dreassi, Elena ; Crespan, E.; Maga, G.; Schenone, S.; Musumeci, F.; Brullo, C.; Richters, A.; Gasparrini, F.; Angelucci, A.; Festuccia, C.; Delle Monache, S.; Rauh, D.; Botta, Maurizio Not applicable
2010Crystal Structure of HIV-1 Reverse Transcriptase Bound to a Non-Nucleoside Inhibitor with a Novel Mechanism of ActionS., Freisz; G., Bec; Radi, Marco; P., Wolff; E., Crespan; Angeli, Lucilla; P., Dumas; G., Maga; Botta, Maurizio ; E., EnnifarNot applicable
2011Design, synthesis, biological activity and ADME properties of pyrazolo[3,4-d]pyrimidines active in hypoxic human leukemia cells: a lead optimization studyRadi, Marco; Dreassi, Elena ; C., Brullo; E., Crespan; Tintori, Cristina; V., Bernardo; Valoti, Massimo; Zamperini, Claudio; H., Daigl; F., Musumeci; Carraro, Fabio; Naldini, Antonella; Filippi, Irene; G., Maga; S., Schenone; Botta, Maurizio Not applicable
2010Dual Src and Abl inhibitors target wild type Abl and the AblT315I Imatinib-resistant mutant with different mechanismE., Crespan; Radi, Marco; S., Zanoli; S., Schenone; Botta, Maurizio ; G., MagaNot applicable
2010HIV-1 RT inhibitors with a novel mechanism of action: NNRTIs that compete with the nucleotide substrateG., Maga; Radi, Marco; M., Gerard; Botta, Maurizio ; E., EnnifarNot applicable
2014Insight into the Allosteric Inhibition of Abl KinaseFallacara, Anna Lucia; Tintori, Cristina; Radi, Marco; Schenone, Silvia; Botta, Maurizio Not applicable
2009Microwave-assisted organocatalytic multicomponent Knoevenagel/Hetero Diels Alder reaction for the synthesis of 2,3-dihydropyran[2,3-c]pyrazolesRadi, Marco; Bernardo, Vincenzo; Bechi, Beatrice; Castagnolo, Daniele; Pagano, Mafalda; Botta, Maurizio Not applicable
2003Microwave-enhanced Sonogashira coupling reaction of substituted pyrimidinones and pyrimidine nucleosidesPetricci, Elena ; Radi, Marco; Corelli, Federico ; Botta, Maurizio Not applicable
2008A Multidisciplinary Approach for the Identification ofNovel HIV-1 Non-Nucleoside Reverse TranscriptaseInhibitors: S-DABOCs and DAVPsRadi, Marco; Falciani, Chiara; Contemori, Lorenzo; Petricci, Elena ; G., Maga; A., Samuele; S., Zanoli; M., Terrazas; Castria, Marinunzia; Togninelli, Andrea; J. A., Esté; I., CLOTET CODINA; M., ARMAND UGON; Botta, Maurizio Not applicable
2010New insights into small-molecule inhibitors of Bcr-AblS., Schenone; Botta, Maurizio ; Radi, Marco; O., BrunoNot applicable
2008A one-pot, two step microwave-assisted synthesis of highly functionalized benzoxazoles using solid-supported reagents (SSRs)Radi, Marco; S., Saletti; Botta, Maurizio Not applicable
2010A Practical One-Pot Two-Step Protocol for the Microwave-Assisted Synthesis of Highly Functionalized Rhodanine DerivativesRadi, Marco; Botta, Lorenzo; Casaluce, Gianni; Bernardini, Martina; Botta, Maurizio Not applicable
2013Pyrazolo[3,4-d]pyrimidine Prodrugs: Strategic Optimization of the Aqueous Solubility of Dual Src/Abl InhibitorsVignaroli, Giulia; Zamperini, Claudio; Dreassi, Elena ; Radi, Marco; Angelucci, A.; Sanità, P.; Crespan, E.; Kissova, M.; Maga, G.; Schenone, S.; Musumeci, F.; Botta, Maurizio Not applicable
2009Recent highlights in the synthesis of highly functionalized pyrimidinesRadi, Marco; Botta, Maurizio ; S., SchenoneNot applicable
2002Solid-phase synthesis (SPS) of substituted uracils via Oxone® cleavage methodologyPetricci, Elena ; Renzulli, MICHELA LUCIA; Radi, Marco; Corelli, Federico ; Botta, Maurizio Not applicable
2008Synthesis of an original oxygenated taxuspine X analogue: a versatile non-natural natural product with remarkable P-gp modulating activityS. I., Avramova; Galletti, Elena; Renzulli, MICHELA LUCIA; Giorgi, Gianluca ; Sgaragli, GIAN PIETRO; Alderighi, Daniela; C., Ghiron; Corelli, Federico ; Radi, Marco; Botta, Maurizio Not applicable
2005Synthesis of reactive cytidine derivatives as building blocks for cross-linking oligonucleotidesRadi, Marco; Mugnaini, Claudia ; Petricci, Elena ; Corelli, Federico ; Botta, Maurizio Not applicable
2013Unconventional Plasticity of HIV-1 Reverse Transcriptase: How Inhibitors Could Open a Connection "Gate" between Allosteric and Catalytic Sites.Bellucci, Luca; Angeli, Lucilla; Tafi, Andrea ; Radi, Marco; Botta, Maurizio Not applicable