Browsing by Author Novellino, E

Showing results 1 to 11 of 11
Issue DateTitleAuthor(s)Third Mission
20111-Aryl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide: An effective scaffold for the design of either CB1 and CB2 receptor ligandsPiscitelli, F; Ligresti, A; LA REGINA, G; Gatti, V; Brizzi, Antonella ; Pasquini, Serena; Allarà, M; CARAI M. A., M; Novellino, E; Colombo, G; DI MARZO, V; Corelli, Federico ; Silvestri, R.Not applicable
2005Development of molecular probes for the identification of extra interaction sites in the mid-gorge and peripheral sites of butyrylcholinesterase (BuChE). Rational design of novel, selective, and highly potent BuChE inhibitors.Campiani, Giuseppe ; Fattorusso, C; Butini, Stefania ; Gaeta, A; Agnusdei, M; Gemma, Sandra ; Persico, M; Catalanotti, B; Savini, Luisa; Nacci, Vito; Novellino, E; Holloway, Hw; Greig, Nh; Belinskaya, T; Fedorko, Jm; Saxena, A.Not applicable
2007Development of piperazine-tethered heterodimers as potent antimalarials against chloroquine-resistant P. falciparum strains. Synthesis and molecular modeling.Gemma, Sandra ; Kukreja, G; Campiani, Giuseppe ; Butini, Stefania ; Bernetti, Matteo; Joshi, Bp; Savini, Luisa; Basilico, N; Taramelli, D; Yardley, V; Bertamino, A; Novellino, E; Persico, M; Catalanotti, B; Fattorusso, C.Not applicable
2010Discovery of Bishomo(hetero)arylpiperazines as Novel Multifunctional Ligands Targeting Dopamine D-3 and Serotonin 5-HT1A and 5-HT2A ReceptorsButini, Stefania ; Campiani, Giuseppe ; Franceschini, Silvia; Trotta, Francesco; Kumar, V; Guarino, Egeria; Borrelli, Giuseppe; Fiorini, Isabella; Novellino, E; Fattorusso, C; Persico, M; Orteca, N; SANDAGER NIELSEN, K; Jacobsen, Ta; Madsen, K; SCHEEL KRUGER, J; Gemma, Sandra Not applicable
2009L-Type calcium channel blockers: from diltiazem to 1,2,4-oxadiazol-5-ones via thiazinooxadiazol-3-one derivatives.Budriesi, R; Cosimelli, B; Ioan, P; Ugenti, Mp; Carosati, E; Frosini, Maria; Fusi, Fabio ; Spisani, R; Saponara, Simona; Cruciani, G; Novellino, E; Spinelli, D; Chiarini, A.Not applicable
2010Malaria chemotherapy: recent advances in drug developmentGemma, Sandra ; Travagli, Valter ; Savini, Luisa; Novellino, E; Campiani, Giuseppe ; Butini, Stefania Not applicable
1999Pyrrolobenzoxazepinone Derivatives as Non-Nucleoside HIV-1 RT Inhibitors: Further Structure-Activity Relationship Studies and Identification of More Potent Broad-Spectrum HIV-1 RT Inhibitors with Antiviral ActivityCampiani, Giuseppe ; Morelli, E; Fabbrini, Monica; Nacci, Vito; Greco, G; Novellino, E; Ramunno, A; Maga, G; Spadari, S; Caliendo, G; Bergamini, A; Faggioli, E; Uccella, I; Bolacchi, F; Marini, S; Coletta, M; Nacca, A; Caccia, S.Not applicable
2005Specific targeting highly conserved residues in the HIV-1 reverse transcriptase primer grip region. Design, synthesis, and biological evaluation of novel, potent, and broad spectrum NNRTIs with antiviral activity.Fattorusso, C; Gemma, Sandra ; Butini, Stefania ; Huleatt, P; Catalanotti, B; Persico, M; DE ANGELIS, M; Fiorini, Isabella; Nacci, Vito; Ramunno, A; Rodriquez, M; Greco, G; Novellino, E; Bergamini, A; Marini, S; Coletta, M; Maga, G; Spadari, S; Campiani, Giuseppe Not applicable
2003Specific targeting of acetylcholinesterase and butyrylcholinesterase recognition sites. Rational design of novel, selective, and highly potent cholinesterase inhibitors.Savini, Luisa; Gaeta, A; Fattorusso, C; Catalanotti, B; Campiani, Giuseppe ; Chiasserini, Luisa ; Pellerano, Cesare; Novellino, E; Mckissic, D; Saxena, A.Not applicable
2013The structural evolution of β-secretase inhibitors: a focus on the development of small-molecule inhibitors.Butini, Stefania ; Brogi, Simone; Novellino, E; Campiani, Giuseppe ; Ghosh, Ak; Brindisi, Margherita ; Gemma, Sandra Not applicable
2010Synthesis of Dihydroplakortin, 6-epi-Dihydroplakortin, and Their C10-Desethyl AnaloguesGemma, Sandra ; Gabellieri, Emanuele; SANNA COCCONE, Salvatore; Marti, F; TAGLIALATELA SCAFATI, O; Novellino, E; Campiani, Giuseppe ; Butini, Stefania Not applicable