Browsing by Author Maga, G


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Issue DateTitleAuthor(s)Third Mission
20093D QSAR models built on structure-based alignments of Abl tyrosine kinase inhibitors.Falchi, F; Manetti, Fabrizio ; Carraro, Fabio; Naldini, Antonella; Maga, G; Crespan, E; Schenone, S; Bruno, O; Brullo, C; Botta, Maurizio Not applicable
2010Design and synthesis of Thiadiazoles and Thiazoles targeting the Bcr-Abl T315I mutant: from docking false positives to ATP-noncompetitive inhibitorsBotta, Maurizio ; Crespan, E; Falchi, F; Bernardo, V; Zanoli, S; Manetti, Fabrizio ; Schenone, S; Maga, G; Botta, Maurizio Not applicable
2009Determination of permeability and lipophilicity of pyrazolo-pyrimidine tyrosine kinase inhibitors and correlation with biological dataDreassi, Elena ; Zizzari, ALESSANDRA TANIA; Falchi, Federico; Schenone, S; Santucci, Annalisa ; Maga, G; Botta, Maurizio Not applicable
2007Dihydro-alkylthio-benzyl-oxopyrimidines as Inhibitors of Reverse Transcriptase: Synthesis and Rationalization of the Biological Data on Both Wild-Type Enzyme and Relevant Clinical MutantsMugnaini, Claudia ; Alongi, M; Togninelli, A; Gevariya, H; Brizzi, Antonella ; Manetti, Fabrizio ; Bernardini, C; Angeli, L; Tafi, Andrea ; Bellucci, L; Corelli, Federico ; Massa, Silvio; Maga, G; Samuele, A; Facchini, M; CLOTET CODINA, I; ARMAND UGON, M; ESTE J., A; Botta, Maurizio Not applicable
2008Discovery and SAR of 1,3,4-thiadiazole derivatives as potent Abl tyrosine kinase inhibitors and cytodifferentiating agentsBotta, Maurizio ; Crespan, E; Botta, G; Falchi, F; Maga, G; Manetti, Fabrizio ; Corradi, V; Mancini, M; SANTUCCI M., A; Schenone, S; Botta, Maurizio Not applicable
2009Discovery of Chiral Cyclopropyl Dihydro-Alkylthio-Benzyl-Oxopyrimidine (S-DABO) Derivatives as Potent HIV-1 Reverse Transcriptase Inhibitors with High Activity Against Clinically Relevant MutantsBotta, Maurizio ; Maga, G; Alongi, M; Angeli, L; Samuele, A; Zanoli, S; Bellucci, L; Tafi, Andrea ; Casaluce, G; Giorgi, Gianluca ; Armand Ugon, M; Gonzalez, E; Esté, Ja; Baltzinger, M; Bec, G; Dumas, P; Ennifar, E; Botta, Maurizio Not applicable
2007Discovery of non-nucleoside inhibitors of HIV-1 reverse transcriptase competing with the nucleotide substrate.Maga, G; Botta, Maurizio ; Zanoli, S; Manetti, Fabrizio ; Cancio, R; Hübscher, U; Spadari, S; Falciani, C; Terrazas, M; Vilarrasa, J; Botta, Maurizio Not applicable
2012Discovery of the first small molecule inhibitor of human DDX3 specifically designed to target the RNA binding site: towards the next generation HIV-1 inhibitorsBotta, Maurizio ; Falchi, F.; Garbelli, A.; Samuele, A.; Bernardo, V.; Paolucci, S.; Baldanti, F.; Schenone, S.; Manetti, Fabrizio ; Maga, G; Botta, Maurizio Not applicable
2007Identification of a novel pyrazolo[3,4-d]pyrimidine able to inhibit cell proliferation of a human osteogenic sarcoma in vitro and in a xenograft model in mice.Manetti, Fabrizio ; Santucci, Annalisa ; Locatelli, Ga; Maga, G; Spreafico, A; Serchi, T; Orlandini, Maurizio ; Bernardini, Giulia ; Caradonna, Np; Spallarossa, A; Brullo, C; Schenone, S; Bruno, O; Ranise, A; Bondavalli, F; Hoffmann, O; Bologna, M; Angelucci, A; Botta, Maurizio Not applicable
2013Identification of Hck inhibitors as hits for the development of antileukemia and anti-HIV agents.Tintori, Cristina; Laurenzana, Ilaria; La Rocca, F; Falchi, Federico; Carraro, Fabio; Ruiz, A; Esté, Ja; Kissova, M; Crespan, E; Maga, G; Biava, M; Brullo, C; Schenone, S; Botta, Maurizio Not applicable
2009Indolyl-pyrrolone as a new scaffold for Pim1 inhibitorsOlla, S; Manetti, Fabrizio ; Crespan, E; Maga, G; Angelucci, A; Schenone, S; Bologna, M; Botta, Maurizio Not applicable
2007Inhibition of Bcr-Abl phosphorylation and induction of apoptosis by pyrazolo[3,4-d] pyrimidines in human leukemia cellsManetti, Fabrizio ; Pucci, Annalisa; Magnani, M; LOCATELLI G., A; Brullo, C; Naldini, Antonella; Schenone, S; Maga, G; Carraro, Fabio; Botta, Maurizio Not applicable
2010Molecular characterization of c-Abl/c-Src kinase inhibitors targeted against murine tumour progenitor cells that express stem cell markers.Kruewel, T; Schenone, S; Botta, Maurizio ; Maga, G; Rohrbeck, A; Botta, M; Borlak, J.Not applicable
2011N-[2-Methyl-5-(triazol-1-yl)phenyl]pyrimidin-2-amine as a scaffold for the synthesis of inhibitors of Bcr-Abl.Arioli, F; Borrelli, S; Colombo, F; Falchi, F; Filippi, Irene; Crespan, E; Naldini, Antonella; Scalia, Giusy; Silvani, A; Maga, G; Carraro, Fabio; Botta, Maurizio ; Passarella, D.Not applicable
2008Pharmacophore modeling and molecular docking led to the discovery of inhibitors of human immunodeficiency virus-1 replication targeting the human cellular aspartic acid-glutamic acid-alanine-aspartic acid box polypeptide 3.Maga, G; Falchi, F; Garbelli, A; Belfiore, A; Witvrouw, M; Manetti, Fabrizio ; Botta, Maurizio Not applicable
2006Pyrazolo[3,4-d]pyrimidines as potent antiproliferative and proapoptotic agents toward A431 and 8701-BC cells in culture via inhibition of c-Src phosphorylation.Carraro, Fabio; Naldini, Antonella; Pucci, Annalisa; Locatelli, Ga; Maga, G; Schenone, S; Bruno, O; Ranise, A; Bondavalli, F; Brullo, C; Fossa, P; Menozzi, G; Mosti, L; Modugno, M; Tintori, Cristina; Manetti, Fabrizio ; Botta, Maurizio Not applicable
1999Pyrrolobenzoxazepinone Derivatives as Non-Nucleoside HIV-1 RT Inhibitors: Further Structure-Activity Relationship Studies and Identification of More Potent Broad-Spectrum HIV-1 RT Inhibitors with Antiviral ActivityCampiani, Giuseppe ; Morelli, E; Fabbrini, Monica; Nacci, Vito; Greco, G; Novellino, E; Ramunno, A; Maga, G; Spadari, S; Caliendo, G; Bergamini, A; Faggioli, E; Uccella, I; Bolacchi, F; Marini, S; Coletta, M; Nacca, A; Caccia, S.Not applicable
2005Specific targeting highly conserved residues in the HIV-1 reverse transcriptase primer grip region. Design, synthesis, and biological evaluation of novel, potent, and broad spectrum NNRTIs with antiviral activity.Fattorusso, C; Gemma, Sandra ; Butini, Stefania ; Huleatt, P; Catalanotti, B; Persico, M; DE ANGELIS, M; Fiorini, Isabella; Nacci, Vito; Ramunno, A; Rodriquez, M; Greco, G; Novellino, E; Bergamini, A; Marini, S; Coletta, M; Maga, G; Spadari, S; Campiani, Giuseppe Not applicable
2008Structure-Based Optimization of Pyrazolo[3,4-d]pyrimidines as Abl Inhibitors and Antiproliferative Agents toward Human Leukemia Cell Lines.Manetti, Fabrizio ; Brullo, C; Magnani, M; Mosci, F; Chelli, B; Crespan, E; Schenone, S; Naldini, Antonella; Bruno, O; Trincavelli, Ml; Maga, G; Carraro, Fabio; Martini, C; Bondavalli, F; Botta, Maurizio Not applicable
2006Synthesis and biological investigation of S-aryl-S-DABO derivatives as HIV-1 inhibitorsMugnaini, Claudia ; Manetti, Fabrizio ; EST J., A; CLOTET CODINA, I; Maga, G; Cancio, R; Botta, Maurizio ; Corelli, Federico Not applicable