Browsing by Author F., Makovec

Showing results 1 to 16 of 16
Issue DateTitleAuthor(s)Third Mission
2007Cyclooxygenase-2 Inhibitors. 1,5-Diarylpyrrol-3-acetic Esters with Enhanced Inhibitory Activity Toward Cyclooxygenase-2 and Improved Cyclooxygenase-2/Cyclooxygenase-1 SelectivityM., Biava; G. C., Porretta; G., Poce; S., Supino; S., Forli; M., Rovini; Cappelli, Andrea ; Manetti, Fabrizio ; Botta, Maurizio ; L., Sautebin; A., Rossi; C., Pergola; C., Ghelardini; E., Vivoli; F., Makovec; P., Anzellotti; P., Patrignani; Anzini, Maurizio Not applicable
2008Design, Synthesis, and Biological Evaluation of AT1 Angiotensin II Receptor Antagonists Based on the Pyrazolo[3,4-b]pyridine and related Heteroaromatic Bicyclic SystemsCappelli, Andrea ; C., Nannicini; A., Gallelli; Giuliani, Germano ; S., Valenti; G., PERICOT MOHR; Anzini, Maurizio ; L., Mennuni; F., Ferrari; G., Caselli; A., Giordani; W., Peris; F., Makovec; Giorgi, Gianluca ; Vomero, SalvatoreNot applicable
2010Design, Synthesis, and Preliminary Biological Evaluation of Pyrrolo[3,4-c]quinolin-1-one and Oxoisoindoline Derivatives as Aggrecanase Inhibitors.Cappelli, Andrea ; C., Nannicini; A. S., Valenti; Giuliani, Germano ; Anzini, Maurizio ; L., Mennuni; A., Giordani; G., Caselli; L. P., Stasi; F., Makovec; Giorgi, Gianluca ; Vomero, SalvatoreNot applicable
2004Design, Synthesis, Structural Studies, Biological Evaluation, and Computational Simulations of Novel Potent AT1 Angiotensin II Receptor Antagonists Based on the 4-Phenylquinoline Structure.Cappelli, Andrea ; G., PERICOT MOHR; A., Gallelli; M., Rizzo; Anzini, Maurizio ; Vomero, Salvatore; L., Mennuni; F., Ferrari; F., Makovec; M. C., Menziani; P. G., DE BENEDETTI; Giorgi, Gianluca Not applicable
2003Determination of a novel angiotensin-AT1 Antagonist CR3210, in biological samples by HPLC.M., Rizzo; Anzini, Maurizio ; Cappelli, Andrea ; Vomero, Salvatore; D., Ventrice; G., DE SARRO; S., Procopio; N., Costa; F., MakovecNot applicable
2003Enzymatic and Molecular Modeling Studies of 5-HT3 Receptor Ligands Based on Pyrroloquinoline Structure and Provided with Acetylcholinesterase Inhibitory ActivityS., Alcaro; F., Ortuso; D., Battaglia; Anzini, Maurizio ; Cappelli, Andrea ; A., Gallelli; G., PERICOT MOHR; Vomero, Salvatore; A., Galli; C., Costagli; F., MakovecNot applicable
2006Further studies on imidazo[4,5-b]pyridine AT1 angiotensin II receptor antagonists. Effects of the transformation of the 4-phenylquinoline backbone into 4-phenylisoquinolinone or 1-phenylindene scaffolds.Cappelli, Andrea ; G., PERICOT MOHR; Giuliani, Germano ; S., Galeazzi; Anzini, Maurizio ; L., Mennuni; F., Ferrari; F., Makovec; E. M., Kleinrath; T., Langer; Valoti, Massimo; Giorgi, Gianluca ; Vomero, SalvatoreNot applicable
2005Further Studies on the Interaction of 5-Hydroxytryptamine3 (5-HT3) Receptor with Arylpiperazine Ligands. Development of a New 5-HT3 Receptor Ligand Showing Potent Acetylcholinesterase Inhibitory Properties.Cappelli, Andrea ; A., Gallelli; M., Manini; Anzini, Maurizio ; L., Mennuni; F., Makovec; M. C., Menziani; S., Alcaro; F., Ortuso; Vomero, SalvatoreNot applicable
2010Multivalent Supramolecular Dendrimer-Based Drugs.S., Galeazzi; T. M., Hermans; Paolino, Marco ; Anzini, Maurizio ; L., Mennuni; A., Giordani; G., Caselli; F., Makovec; E. W., Meijer; Vomero, Salvatore; Cappelli, Andrea Not applicable
2010Novel Ester and Acid Derivatives of the 1,5-Diarylpyrrole Scaffold as Anti-inflammatory and Analgesic Agents. Synthesis, in vitro and in vivo Biological Evaluation.M., Biava; G. C., Porretta; G., Poce; C., Battilocchio; Manetti, Fabrizio ; Botta, Maurizio ; S., Forli; L., Sautebin; A., Rossi; C., Pergola; C., Ghelardini; N., Galeotti; F., Makovec; A., Giordani; P., Anzellotti; P., Patrignani; Anzini, Maurizio Not applicable
1999Novel Potent and Selective Central 5-HT3 Receptor Ligands Provided with Different Intrinsic Efficacy. 2. Molecular Basis of the Intrinsic Efficacy of Arylpiperazine Derivatives at the Central 5-HT3 ReceptorsCappelli, Andrea ; Anzini, Maurizio ; Vomero, Salvatore; L., Canullo; L., Mennuni; F., Makovec; E., Doucet; M., Hamon; M. C., Menziani; P. G., DE BENEDETTI; G., Bruni; M. R., Romeo; Giorgi, Gianluca ; Donati, Alessandro Not applicable
1998Novel potent and selective central 5-HT3 receptor ligands provided with different intrinsic efficacy. I. Mapping the central 5-HT3 recceptor binding site by arylpiperazine derivativesCappelli, Andrea ; Anzini, Maurizio ; Vomero, Salvatore; L., Mennuni; F., Makovec; E., Doucet; M., Hamon; G., Bruni; M. R., Romeo; M. C., Menziani; P. G., DE BENEDETTI; T., LangerNot applicable
2004Sensitive SPE-HPLC Method to Determine a Novel Angiotensin-AT1 Antagonist in Biological Samples.M., Rizzo; D., Ventrice; F., Monforte; S., Procopio; G., DE SARRO; Anzini, Maurizio ; Cappelli, Andrea ; F., MakovecNot applicable
2005Structure–affinity relationship studies on arylpiperazine derivatives related to quipazine as serotonin transporter ligands. Molecular basis of the selectivity SERT/5-HT3 receptor.Cappelli, Andrea ; Giuliani, Germano ; A., Gallelli; S., Valenti; Anzini, Maurizio ; L., Mennuni; F., Makovec; A., Cupello; Vomero, SalvatoreNot applicable
2003Synthesis and Characterization of a New Benzofulvene Polymer Showing a Thermoreversible Polymerization BehaviorCappelli, Andrea ; G., PERICOT MOHR; Anzini, Maurizio ; Vomero, Salvatore; Donati, Alessandro ; Casolaro, Mario ; R., Mendichi; Giorgi, Gianluca ; F., MakovecNot applicable
2011Synthesis and Structure-Activity Relationship Studies in Translocator Protein Ligands Based on a Pyrazolo[3,4-b]quinoline ScaffoldCappelli, Andrea ; G., Bini; S., Valenti; Giuliani, Germano ; Paolino, Marco ; Anzini, Maurizio ; Vomero, Salvatore; Giorgi, Gianluca ; A., Giordani; L. P., Stasi; F., Makovec; C., Ghelardini; L., DI CESARE MANNELLI; A., Concas; P., Porcu; G., BiggioNot applicable