Browsing by Author E., Crespan

Showing results 1 to 6 of 6
Issue DateTitleAuthor(s)Third Mission
2010Crystal Structure of HIV-1 Reverse Transcriptase Bound to a Non-Nucleoside Inhibitor with a Novel Mechanism of ActionS., Freisz; G., Bec; Radi, Marco; P., Wolff; E., Crespan; Angeli, Lucilla; P., Dumas; G., Maga; Botta, Maurizio ; E., EnnifarNot applicable
2011Design, synthesis, biological activity and ADME properties of pyrazolo[3,4-d]pyrimidines active in hypoxic human leukemia cells: a lead optimization studyRadi, Marco; Dreassi, Elena ; C., Brullo; E., Crespan; Tintori, Cristina; V., Bernardo; Valoti, Massimo; Zamperini, Claudio; H., Daigl; F., Musumeci; Carraro, Fabio; Naldini, Antonella; Filippi, Irene; G., Maga; S., Schenone; Botta, Maurizio Not applicable
2010Dual Src and Abl inhibitors target wild type Abl and the AblT315I Imatinib-resistant mutant with different mechanismE., Crespan; Radi, Marco; S., Zanoli; S., Schenone; Botta, Maurizio ; G., MagaNot applicable
2008N-(thiazol-2-yl)-2-thiophene carboxamide derivatives as Abl inhibitors identified by a pharmacophore-based database screening of commercially available compoundsManetti, Fabrizio ; F., Falchi; E., Crespan; S., Schenone; G., Maga; Botta, Maurizio Not applicable
2005Parallel Solution-Phase and Microwave-Assisted Synthesis of New S-DABO Derivatives Endowed with Subnanomolar Anti-HIV-1 ActivityManetti, Fabrizio ; J. A., Este; I., CLOTET CODINA; M., ARMAND UGON; G., Maga; E., Crespan; R., Cancio; Mugnaini, Claudia ; C., Bernardini; A., Togninelli; C., Carmi; M., Alongi; Petricci, Elena ; S., Massa; Corelli, Federico ; Botta, Maurizio Not applicable
2008Selective targeting of the HIV-1 reverse transcriptase catalytic complex through interaction with the ‘‘primer grip’’ region by pyrrolobenzoxazepinone non-nucleoside inhibitors correlates with increased activity towards drug-resistant mutants.S., Zanoli; Gemma, Sandra ; Butini, Stefania ; Brindisi, Margherita ; B. P., Joshi; Campiani, Giuseppe ; C., Fattorusso; M., Persico; E., Crespan; R., Cancio; S., Spadari; U., Hubscher; G., MagaNot applicable