Browsing by Author Docquier, J. D.

Showing results 1 to 7 of 7
Issue DateTitleAuthor(s)Third Mission
20204-(N-alkyl-and-acyl-amino)-1,2,4-triazole-3-thione analogs as metallo-β-lactamase inhibitors: Impact of 4-linker on potency and spectrum of inhibitionGavara, L.; Verdirosa, F.; Legru, A.; Mercuri, P. S.; Nauton, L.; Sevaille, L.; Feller, G.; Berthomieu, D.; Sannio, F.; Marcoccia, F.; Tanfoni, S.; Luca, F. D.; Gresh, N.; Galleni, M.; Docquier, J. D.; Hernandez, J. -F.Not applicable
2020ANT2681: SAR Studies Leading to the Identification of a Metallo-β-lactamase Inhibitor with Potential for Clinical Use in Combination with Meropenem for the Treatment of Infections Caused by NDM-Producing EnterobacteriaceaeDavies, D. T.; Leiris, S.; Sprynski, N.; Castandet, J.; Lozano, C.; Bousquet, J.; Zalacain, M.; Vasa, S.; Dasari, P. K.; Pattipati, R.; Vempala, N.; Gujjewar, S.; Godi, S.; Jallala, R.; Sathyap, R. R.; Darshanoju, N. A.; Ravu, V. R.; Juventhala, R. R.; Pottabathini, N.; Sharma, S.; Pothukanuri, S.; Holden, K.; Warn, P.; Marcoccia, F.; Benvenuti, Manuela ; Pozzi, Cecilia ; Mangani, Stefano ; Docquier, J. D.; Lemonnier, M.; Everett, M.Not applicable
2020Discovery of ANT3310, a Novel Broad-Spectrum Serine β-Lactamase Inhibitor of the Diazabicyclooctane Class, Which Strongly Potentiates Meropenem Activity against Carbapenem-Resistant Enterobacterales and Acinetobacter baumanniiDavies, D. T.; Leiris, S.; Zalacain, M.; Sprynski, N.; Castandet, J.; Bousquet, J.; Lozano, C.; Llanos, A.; Alibaud, L.; Vasa, S.; Pattipati, R.; Valige, R.; Kummari, B.; Pothukanuri, S.; De Piano, C.; Morrissey, I.; Holden, K.; Warn, P.; Marcoccia, F.; Benvenuti, Manuela ; Pozzi, Cecilia ; Tassone, Giusy ; Mangani, Stefano ; Docquier, J. D.; Pallin, D.; Elliot, R.; Lemonnier, M.; Everett, M.Not applicable
2020Discovery of Taniborbactam (VNRX-5133): A Broad-Spectrum Serine- And Metallo-β-lactamase Inhibitor for Carbapenem-Resistant Bacterial InfectionsLiu, B.; Trout, R. E. L.; Chu, G. -H.; Mcgarry, D.; Jackson, R. W.; Hamrick, J. C.; Daigle, D. M.; Cusick, S. M.; Pozzi, Cecilia ; De Luca, F.; Benvenuti, Manuela ; Mangani, Stefano ; Docquier, J. D.; Weiss, W. J.; Pevear, D. C.; Xerri, L.; Burns, C. J.Not applicable
2017Identification, synthesis and biological activity of alkyl-guanidine oligomers as potent antibacterial agentsZamperini, C.; Maccari, G.; Deodato, D.; Pasero, Carolina; D'Agostino, Ilaria ; Orofino, Francesco ; De Luca, F.; Dreassi, Elena ; Docquier, J. D.; Botta, Maurizio Not applicable
2020Virtual screening identifies broad-spectrum β-lactamase inhibitors with activity on clinically relevant serine- and metallo-carbapenemasesSpyrakis, F.; Santucci, M.; Maso, L.; Cross, S.; Gianquinto, E.; Sannio, F.; Verdirosa, F.; De Luca, F.; Docquier, J. D.; Cendron, L.; Tondi, D.; Venturelli, A.; Cruciani, G.; Costi, M. P.Not applicable
2020VNRX-5133 (Taniborbactam), a broad-spectrum inhibitor of serine- And metallo-β-lactamases, restores activity of cefepime in enterobacterales and Pseudomonas aeruginosaHamrick, J. C.; Docquier, J. D.; Uehara, T.; Myers, C. L.; Six, D. A.; Chatwin, C. L.; John, K. J.; Vernacchio, S. F.; Cusick, S. M.; Trout, R. E. L.; Pozzi, Cecilia ; De Luca, F.; Benvenuti, Manuela ; Mangani, Stefano ; Liu, B.; Jackson, R. W.; Moeck, G.; Xerri, L.; Burns, C. J.; Pevear, D. C.; Daigle, D. M.Not applicable