Browsing by Author C., Fattorusso

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Issue DateTitleAuthor(s)Third Mission
2001Characterisation of 1H-cyclopentapyrimidine-2,4(1H,3H)-dione derivative (S)-CPW399 as a novel, potent and subtype-selective AMPA receptor full agonist with partial desensitization propertiesCampiani, Giuseppe ; E., Morelli; Nacci, Vito; C., Fattorusso; A., Ramunno; E., Novellino; J., Greenwood; T., Liljefors; R., Griffiths; C., Sinclair; H., Reavy; A. S., Kristensen; D. S., Pickering; A., Schousboe; A., Cagnotto; E., Fumagalli; T., MenniniNot applicable
2009Combining 4-Aminoquinoline- and Clotrimazole-based Pharmacophores towards Innovative and Potent Hybrid Antimalarials.Gemma, Sandra ; Campiani, Giuseppe ; Butini, Stefania ; B. P., Joshi; G., Kukreja; SANNA COCCONE, Salvatore; Bernetti, Matteo; M., Persico; Nacci, Vito; Fiorini, Isabella; E., Novellino; D., Taramelli; N., Basilico; S., Parapini; V., Yardley; S., Croft; S., KELLER MAERKI; M., Rottmann; R., Brun; M., Coletta; S., Marini; G., Guiso; S., Caccia; C., FattorussoNot applicable
2006Conformational Flexibility in the Peripheral Site of Torpedo californica Acetylcholinesterase Revealed by the Complex Structure with a Bifunctional InhibitorJ. P., Colletier; B., Sanson; F., Nachon; E., Gabellieri; C., Fattorusso; M., Weik; Campiani, Giuseppe Not applicable
2007Design and Synthesis of Potent Antimalarial Agents Based on Clotrimazole Scaffold: Exploring an Innovative Pharmacophore.Gemma, Sandra ; Campiani, Giuseppe ; Butini, Stefania ; B., Joshi; G., Kukreja; M., Persico; B., Catalanotti; E., Novellino; Fattorusso, E; Nacci, Vito; Savini, Luisa; D., Taramelli; N., Basilico; G., Morace; V., Yardley; C., FattorussoNot applicable
2008Design, synthesis, and structure-activity relationship studies of 4-quinolinyl- and 9-acrydinylhydrazones as potent antimalarial agents.C., Fattorusso; Campiani, Giuseppe ; G., Kukreja; M., Persico; Butini, Stefania ; Romano, MARIA PIA; Altarelli, Maria; S., Ros; Brindisi, Margherita ; Savini, Luisa; E., Novellino; Nacci, Vito; E., Fattorusso; S., Parapini; N., Basilico; D., Taramelli; V., Yardley; S., Croft; M., Borriello; Gemma, Sandra Not applicable
2006Discovery of Huperzine A/Tacrine Hybrids as Potent Inhibitors of Human Cholinesterases Targeting Their Mid-gorge Recognition SitesGemma, Sandra ; Gabellieri, Emanuele; Huleatt, P.; C., Fattorusso; M., Borriello; B., Catalanotti; Butini, Stefania ; M., DE ANGELIS; E., Novellino; Nacci, Vito; T., Belinskaya; Saxena, Ashima; Campiani, Giuseppe Not applicable
2006Endoperoxide Derivatives from Marine Organisms: 1,2-Dioxanes of the Plakortin Family as Novel Antimalarial AgentsC., Fattorusso; Campiani, Giuseppe ; B., Catalanotti; M., Persico; N., Basilico; S., Parapini; D., Taramelli; C., Campagnuolo; Fattorusso, E; A., Romano; O., TAGLIALATELA SCAFATINot applicable
2008Exploiting Protein Fluctuations at the Active-Site Gorge of Human Cholinesterases: Further Optimization of the Design Strategy to Develop Extremely Potent InhibitorsButini, Stefania ; Campiani, Giuseppe ; M., Borriello; Gemma, Sandra ; Panico, Alessandro; M., Persico; B., Catalanotti; S., Ros; Brindisi, Margherita ; M., Agnusdei; Fiorini, Isabella; Nacci, Vito; E., Novellino; T., Belinskaya; A., Saxena; C., FattorussoNot applicable
2008Microwave-assisted synthesis of 4-quinolylhydrazines followed by nickel boride reduction: a convenient approach to 4-aminoquinolines and derivativesGemma, Sandra ; G., Kukreja; Tripaldi, Pierangela; Altarelli, Maria; Bernetti, Matteo; Franceschini, Silvia; Savini, Luisa; Campiani, Giuseppe ; C., Fattorusso; Butini, Stefania Not applicable
2002Non-Nucleoside HIV-1 Reverse Transcriptase (RT) Inhibitors: Past, Present, and Future PerspectivesCampiani, Giuseppe ; A., Ramunno; G., Maga; Nacci, Vito; C., Fattorusso; B., Catalanotti; E., Morelli; E., NovellinoNot applicable
2001Novel and potent tacrine-related hetero- and homobivalent ligands for acetylcholinesterase and butyrylcholinesteraseSavini, Luisa; Campiani, Giuseppe ; A., Gaeta; Pellerano, Cesare; C., Fattorusso; Chiasserini, Luisa ; J. M., Fedorko; A., SaxenaNot applicable
2003Novel antipsychotic agents: recent advances in the drug treatment of schizophreniaButini, Stefania ; Campiani, Giuseppe ; M., DE ANGELIS; C., Fattorusso; Nacci, Vito; Fiorini, IsabellaNot applicable
2005Novel atypical antipsychotic agents: rational design, an efficient palladium-catalyzed route, and pharmacological studiesCampiani, Giuseppe ; Butini, Stefania ; C., Fattorusso; F., Trotta; Gemma, Sandra ; B., Catalanotti; Nacci, Vito; Fiorini, Isabella; A., Cagnotto; I., Mereghetti; T., Mennini; P., Minetti; M. A., DI CESARE; M. A., Stasi; S., DI SERIO; O., Ghirardi; O., Tinti; P., CarminatiNot applicable
2003“A palladium-catalyzed synthetic approach to new Huperzine A analogues modified at the pyridone ring”Gemma, Sandra ; Butini, Stefania ; C., Fattorusso; Fiorini, Isabella; Nacci, Vito; K., Bellebaum; D., Mckissic; A., Saxena; Campiani, Giuseppe Not applicable
2002Pyrrolo 1,3 benzothiazepine-based Atypical Antipsychotic Agents. Synthesis, Structure-Activity Relationship, Molecular Modeling, and Biological StudiesCampiani, Giuseppe ; Butini, Stefania ; Gemma, Sandra ; Nacci, Vito; C., Fattorusso; B., Catalanotti; Giorgi, Gianluca ; A., Cagnotto; M., Goegan; T., Mennini; P., Minetti; L., DI CESARE MANNELLI; D., Mastroianni; N., Scafetta; B., Galletti; M., Stasi; M., Castorina; L., Pacifici; O., Ghirardi; O., Tinti; P., CarminatiNot applicable
2001Pyrrolo-1,5-benzoxazepines Induce Apoptosis in Chronic Myelogenous Leukemia Cells (CML) by Bypassing the Apoptotic Suppressor Bcr-AblM., Mcgee; Campiani, Giuseppe ; A., Ramunno; C., Fattorusso; Nacci, Vito; M., Lawler; D. C., Williams; D. M., ZistererNot applicable
2001Pyrrolo-1,5-benzoxazepines: a new class of apoptotic agentsD. M., Zisterer; M. M., Mcgee; Campiani, Giuseppe ; A., Ramunno; C., Fattorusso; Nacci, Vito; M., Lawler; D. C., WilliamsNot applicable
2005Pyrrolo[1,5]benzoxa(thia)zepines as a New Class of Potent Apoptotic Agents. Biological Studies and Identification of an Intracellular Location of Their Drug TargetM. M., MC GEE; Gemma, Sandra ; Butini, Stefania ; A., Ramunno; D. M., Zisterer; C., Fattorusso; B., Catalanotti; G., Kukreja; Fiorini, Isabella; C., Pisano; C., Cucco; E., Novellino; Nacci, Vito; D. C., Williams; Campiani, Giuseppe Not applicable
2001A rational approach to the design of selective substrates and potent non-transportable inhibitors of the excitatory amino acid transporter EAAC1 (EAAT3). New glutamate and aspartate analogues as potential neuroprotective agents.Campiani, Giuseppe ; M., De Angelis; S., Armaroli; C., Fattorusso; B., Catalanotti; A., Ramunno; Nacci, Vito; E., Novellino; C., Grewer; D., Ionescu; T., Rauen; R., Griffiths; C., Sinclair; E., Fumagalli; T., MenniniNot applicable
2008Selective targeting of the HIV-1 reverse transcriptase catalytic complex through interaction with the ‘‘primer grip’’ region by pyrrolobenzoxazepinone non-nucleoside inhibitors correlates with increased activity towards drug-resistant mutants.S., Zanoli; Gemma, Sandra ; Butini, Stefania ; Brindisi, Margherita ; B. P., Joshi; Campiani, Giuseppe ; C., Fattorusso; M., Persico; E., Crespan; R., Cancio; S., Spadari; U., Hubscher; G., MagaNot applicable